NZ244896A - Quinoxaline-carboxylic and -phosphonic acid derivatives and pharmaceutical compositions - Google Patents
Quinoxaline-carboxylic and -phosphonic acid derivatives and pharmaceutical compositionsInfo
- Publication number
- NZ244896A NZ244896A NZ244896A NZ24489692A NZ244896A NZ 244896 A NZ244896 A NZ 244896A NZ 244896 A NZ244896 A NZ 244896A NZ 24489692 A NZ24489692 A NZ 24489692A NZ 244896 A NZ244896 A NZ 244896A
- Authority
- NZ
- New Zealand
- Prior art keywords
- acid
- dioxo
- tetrahydroquinoxalin
- nitro
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6509—Six-membered rings
- C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
- C07F9/650994—Six-membered rings having the nitrogen atoms in the positions 1 and 4 condensed with carbocyclic rings or carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
- C07D241/40—Benzopyrazines
- C07D241/44—Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Biochemistry (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Psychology (AREA)
- Endocrinology (AREA)
- Molecular Biology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Otolaryngology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4135871A DE4135871A1 (de) | 1991-10-26 | 1991-10-26 | Chinoxalinderivate, deren herstellung und verwendung in arzneimitteln |
| DE4224200 | 1992-07-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ244896A true NZ244896A (en) | 1995-07-26 |
Family
ID=25908683
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ244896A NZ244896A (en) | 1991-10-26 | 1992-10-27 | Quinoxaline-carboxylic and -phosphonic acid derivatives and pharmaceutical compositions |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0565683A1 (fr) |
| JP (1) | JP3258008B2 (fr) |
| KR (1) | KR100262371B1 (fr) |
| CN (1) | CN1038840C (fr) |
| AU (1) | AU664212B2 (fr) |
| CA (1) | CA2099270A1 (fr) |
| CZ (1) | CZ286351B6 (fr) |
| FI (1) | FI932959A0 (fr) |
| HU (1) | HUT64756A (fr) |
| IL (1) | IL103538A (fr) |
| NO (1) | NO304693B1 (fr) |
| NZ (1) | NZ244896A (fr) |
| PL (1) | PL171125B1 (fr) |
| PT (1) | PT101004B (fr) |
| RU (1) | RU2117663C1 (fr) |
| SK (1) | SK281518B6 (fr) |
| WO (1) | WO1993008173A1 (fr) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK162491D0 (da) * | 1991-09-20 | 1991-09-20 | Novo Nordisk As | Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne |
| AU672617B2 (en) * | 1992-06-22 | 1996-10-10 | Regents Of The University Of California, The | Glycine receptor antagonists and the use thereof |
| DE4314592A1 (de) * | 1993-04-28 | 1994-11-03 | Schering Ag | Benzo(f)chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| IL109397A0 (en) | 1993-04-28 | 1994-07-31 | Schering Ag | Quinoxalinedione derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same |
| DE4428152A1 (de) * | 1994-06-22 | 1996-01-04 | Basf Ag | Neue Amido-chinoxalindione, ihrer Herstellung und Verwendung |
| GB9419318D0 (en) * | 1994-09-24 | 1994-11-09 | Pfizer Ltd | Therapeutic agents |
| CN1067387C (zh) * | 1994-09-27 | 2001-06-20 | 山之内制药株式会社 | 1,2,3,4-四氢喹喔啉二酮衍生物 |
| DE4439493A1 (de) * | 1994-10-25 | 1996-05-02 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| DE4439492A1 (de) * | 1994-10-25 | 1996-05-02 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| US6110911A (en) * | 1995-06-07 | 2000-08-29 | Warner-Lambert Company | Cyclic amine derivatives of substituted quinoxaline 2,3-diones as glutamate receptor antagonists |
| DE19521058A1 (de) * | 1995-06-09 | 1996-12-12 | Basf Ag | Verfahren zur Herstellung von Aromaten enthaltenden Polyetherpolyolen |
| DE19545251A1 (de) * | 1995-11-24 | 1997-05-28 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| TW448171B (en) * | 1996-06-06 | 2001-08-01 | Yamanouchi Pharma Co Ltd | Imidazole-substituted quinoxalinedione derivatives |
| DE19624808A1 (de) | 1996-06-21 | 1998-01-02 | Basf Ag | Pyrrolylchinoxalindione, ihre Herstellung und Verwendung |
| DE19728326A1 (de) * | 1997-06-27 | 1999-01-07 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| US6015800A (en) * | 1997-09-03 | 2000-01-18 | Warner-Lambert Company | Substituted quinoxaline-2-ones as glutamate receptor antagonists |
| IL125950A0 (en) * | 1997-09-05 | 1999-04-11 | Pfizer Prod Inc | Methods of administering ampa receptor antagonists to treat dyskinesias associated with dopamine agonist therapy |
| EP0900567A3 (fr) * | 1997-09-05 | 2001-05-02 | Pfizer Products Inc. | Quinazoline-4-ones antagonistes d'AMPA pour le traitement des dyscinésies associées à la thérapie aux agonistes de la dopamine |
| FR2769309B1 (fr) | 1997-10-08 | 2001-06-15 | Oreal | Composition de teinture d'oxydation des fibres keratiniques comprenant un derive d'aminoacide en tant que base d'oxydation et nouveaux derives d'aminoacides |
| JP3790704B2 (ja) | 2001-12-18 | 2006-06-28 | 三菱電機株式会社 | 高周波信号用トランジスタの位相調整回路、及び、半導体集積回路 |
| GB0311406D0 (en) * | 2003-05-17 | 2003-06-25 | Queen Mary & Westfield College | Substituted phosphonate fluorescent sensors,and use thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0118982A1 (fr) * | 1983-02-01 | 1984-09-19 | Sumitomo Chemical Company, Limited | Composés organo-phosphorés de la quinoxalinone, leur production et utilisation |
| NO179551C (no) * | 1987-11-10 | 1996-10-30 | Novo Nordisk As | Analogifremgangsmåte for fremstilling av terapeutisk virksomme kinoxalinforbindelser |
| DK69790D0 (da) * | 1990-03-16 | 1990-03-16 | Novo Nordisk As | Heterocykliske forbindelser, deres fremstilling af anvendelse |
-
1992
- 1992-10-23 PT PT101004A patent/PT101004B/pt not_active IP Right Cessation
- 1992-10-25 JP JP50735393A patent/JP3258008B2/ja not_active Expired - Fee Related
- 1992-10-25 RU RU93044489A patent/RU2117663C1/ru active
- 1992-10-25 KR KR1019930701948A patent/KR100262371B1/ko not_active Expired - Fee Related
- 1992-10-25 SK SK727-93A patent/SK281518B6/sk unknown
- 1992-10-25 PL PL92299929A patent/PL171125B1/pl unknown
- 1992-10-25 HU HU9301877A patent/HUT64756A/hu unknown
- 1992-10-25 WO PCT/DE1992/000895 patent/WO1993008173A1/fr not_active Application Discontinuation
- 1992-10-25 CA CA002099270A patent/CA2099270A1/fr not_active Abandoned
- 1992-10-25 EP EP92922676A patent/EP0565683A1/fr not_active Withdrawn
- 1992-10-25 AU AU28894/92A patent/AU664212B2/en not_active Ceased
- 1992-10-25 IL IL10353892A patent/IL103538A/en not_active IP Right Cessation
- 1992-10-25 CZ CZ19931387A patent/CZ286351B6/cs not_active IP Right Cessation
- 1992-10-26 CN CN92113338A patent/CN1038840C/zh not_active Expired - Fee Related
- 1992-10-27 NZ NZ244896A patent/NZ244896A/en unknown
-
1993
- 1993-06-24 FI FI932959A patent/FI932959A0/fi unknown
- 1993-06-25 NO NO932116A patent/NO304693B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP3258008B2 (ja) | 2002-02-18 |
| CA2099270A1 (fr) | 1993-04-27 |
| PT101004B (pt) | 1999-10-29 |
| NO304693B1 (no) | 1999-02-01 |
| PL299929A1 (en) | 1994-04-05 |
| HUT64756A (en) | 1994-02-28 |
| FI932959A7 (fi) | 1993-06-24 |
| KR100262371B1 (ko) | 2000-08-01 |
| NO932344D0 (no) | 1993-06-25 |
| RU2117663C1 (ru) | 1998-08-20 |
| AU664212B2 (en) | 1995-11-09 |
| JPH06503583A (ja) | 1994-04-21 |
| NO932344L (no) | 1993-06-25 |
| SK281518B6 (sk) | 2001-04-09 |
| HU9301877D0 (en) | 1993-09-28 |
| CN1072929A (zh) | 1993-06-09 |
| EP0565683A1 (fr) | 1993-10-20 |
| CZ138793A3 (en) | 1994-01-19 |
| PT101004A (pt) | 1994-01-31 |
| CN1038840C (zh) | 1998-06-24 |
| PL171125B1 (pl) | 1997-03-28 |
| SK72793A3 (en) | 1993-10-06 |
| CZ286351B6 (cs) | 2000-03-15 |
| WO1993008173A1 (fr) | 1993-04-29 |
| AU2889492A (en) | 1993-05-21 |
| IL103538A (en) | 2001-07-24 |
| KR930703271A (ko) | 1993-11-29 |
| FI932959A0 (fi) | 1993-06-24 |
| IL103538A0 (en) | 1993-03-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NZ244896A (en) | Quinoxaline-carboxylic and -phosphonic acid derivatives and pharmaceutical compositions | |
| KR970011279B1 (ko) | 퀴녹살린 화합물, 이의 제조방법 및 이를 함유하는 약제학적 조성물 | |
| JP2550456B2 (ja) | 縮合ピラジン誘導体 | |
| US5977107A (en) | Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonists | |
| US6143733A (en) | Quinoxalinedione derivatives, their production and use in pharmaceutical agents | |
| EP0676397B1 (fr) | Dérivés d'oxopyridylquinoxaline | |
| JPH0532391B2 (fr) | ||
| US6057304A (en) | Quinoxaline-phosphonic acid derivatives | |
| US6486143B2 (en) | 6-amino- or 6-hydrazino-sulphonyl-3-quinolynyl-phosphonic acid compounds | |
| US6420386B1 (en) | Aryl or heteroaryl quinolylphosphonic acid compounds | |
| PL174418B1 (pl) | Nowe związki, pochodne pirydo [1,2,3-de] chinoksaliny i sposób wytwarzania nowych związków, pochodnych pirydo [1,2,3-de] chinoksaliny | |
| WO1996008492A1 (fr) | DERIVES DE LA [1,2,4]TRIAZOLO[4,3-a]QUINOXALINONE, LEUR PREPARATION ET UTILISATION | |
| DE4314592A1 (de) | Benzo(f)chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln | |
| JPH10506620A (ja) | 〔1,2,4〕トリアゾロ〔4,3−a〕キノキサリノン誘導体、それらの調製方法及び使用 | |
| JP2889150B2 (ja) | オキソピリジニルキノキサリン誘導体 | |
| HUP0100750A2 (hu) | Új 6-szulfamoil-3-kinolilfoszfonsav származékok, eljárás előállításukra és ilyen vegyületeket tartalmazó gyógyszerkészítmények | |
| JPH0859660A (ja) | グルタミン酸受容体拮抗作用を有するアリールチオキノキサリン誘導体 |