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AU2001264595A1 - Sulfonamide and carbamide derivatives of 6(5h)phenanthridinones and their uses - Google Patents

Sulfonamide and carbamide derivatives of 6(5h)phenanthridinones and their uses

Info

Publication number
AU2001264595A1
AU2001264595A1 AU2001264595A AU6459501A AU2001264595A1 AU 2001264595 A1 AU2001264595 A1 AU 2001264595A1 AU 2001264595 A AU2001264595 A AU 2001264595A AU 6459501 A AU6459501 A AU 6459501A AU 2001264595 A1 AU2001264595 A1 AU 2001264595A1
Authority
AU
Australia
Prior art keywords
phenanthridinones
sulfonamide
carbamide derivatives
carbamide
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001264595A
Other languages
English (en)
Inventor
Dana V. Ferraris
Vincent J Kalish
Paul W. Kletzly
Jia-He Li
Larisa E. Serdyuk
Ge Xiao
Jie Zhang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai Corp of North America
Original Assignee
Guilford Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Guilford Pharmaceuticals Inc filed Critical Guilford Pharmaceuticals Inc
Publication of AU2001264595A1 publication Critical patent/AU2001264595A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/10—Aza-phenanthrenes
    • C07D221/12—Phenanthridines

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2001264595A 2000-05-19 2001-05-15 Sulfonamide and carbamide derivatives of 6(5h)phenanthridinones and their uses Abandoned AU2001264595A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20525900P 2000-05-19 2000-05-19
US60205259 2000-05-19
PCT/US2001/015571 WO2001090077A1 (fr) 2000-05-19 2001-05-15 Derives de sulfonamide et de carbamide de 6(5h) phenanthridinones et utilisations de ceux-ci

Publications (1)

Publication Number Publication Date
AU2001264595A1 true AU2001264595A1 (en) 2001-12-03

Family

ID=22761477

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001264595A Abandoned AU2001264595A1 (en) 2000-05-19 2001-05-15 Sulfonamide and carbamide derivatives of 6(5h)phenanthridinones and their uses

Country Status (3)

Country Link
US (1) US6723733B2 (fr)
AU (1) AU2001264595A1 (fr)
WO (1) WO2001090077A1 (fr)

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