BE759493A - Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer - Google Patents
Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquerInfo
- Publication number
- BE759493A BE759493A BE759493DA BE759493A BE 759493 A BE759493 A BE 759493A BE 759493D A BE759493D A BE 759493DA BE 759493 A BE759493 A BE 759493A
- Authority
- BE
- Belgium
- Prior art keywords
- thieno
- pyrimidines
- furyl
- news
- nitro
- Prior art date
Links
- -1 5-NITRO-2-FURYL Chemical class 0.000 title 1
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19691959403 DE1959403A1 (de) | 1969-11-26 | 1969-11-26 | Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
| DE19702050816 DE2050816A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
| DE19702050815 DE2050815A1 (de) | 1970-10-16 | 1970-10-16 | Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine |
| DE19702050814 DE2050814A1 (de) | 1970-10-16 | 1970-10-16 | Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE759493A true BE759493A (fr) | 1971-05-25 |
Family
ID=27430978
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE759493D BE759493A (fr) | 1969-11-26 | Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US3661908A (fr) |
| BE (1) | BE759493A (fr) |
| BG (2) | BG17799A3 (fr) |
| CA (1) | CA926865A (fr) |
| CH (3) | CH559210A5 (fr) |
| DK (1) | DK128781B (fr) |
| FR (1) | FR2073416B1 (fr) |
| GB (1) | GB1321316A (fr) |
| IE (1) | IE34765B1 (fr) |
| IL (1) | IL35729A (fr) |
| NL (1) | NL7017210A (fr) |
| NO (1) | NO129954B (fr) |
| SE (1) | SE377938B (fr) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3932642A (en) * | 1971-04-10 | 1976-01-13 | Boehringer Ingelheim Gmbh | Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use |
| US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| US6608053B2 (en) * | 2000-04-27 | 2003-08-19 | Yamanouchi Pharmaceutical Co., Ltd. | Fused heteroaryl derivatives |
| US20040138238A1 (en) * | 2002-08-08 | 2004-07-15 | Dhanoa Dale S. | Substituted aminopyrimidine compounds as neurokinin antagonists |
| GB0423653D0 (en) * | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
| PT2024372E (pt) | 2006-04-26 | 2010-09-16 | Hoffmann La Roche | Derivado de tieno[3,2-d]pirimidina útil como inibidor de pi3k |
| BRPI0710908A2 (pt) | 2006-04-26 | 2012-06-26 | Genentech Inc | compostos inibidores de fosfoinositìdeo 3-cinase e composições farmacêuticas contendo-os |
| BRPI0710943A2 (pt) * | 2006-04-26 | 2012-06-26 | Genentech Inc | compostos farmacêuticos |
| BRPI0717907A2 (pt) * | 2006-12-07 | 2013-11-05 | Genentech Inc | "composto, composição farmacêutica, métodos para tratar um câncer, para inbir ou modular a atividade da lipídeo quinase, processo para a produçãoo de uma composição farmacêutica, uso de um composto e kit" |
| CL2007003520A1 (es) * | 2006-12-07 | 2008-08-22 | Piramed Ltd Genentech Inc | Compuestos derivados de heterociclos sustituidos con morfolina, inhibidores de la actividad pi3 quinasa; composicion farmaceutica que comprende a dichos compuestos; kit farmaceutico; y su uso para el tratamiento profilactico o terapeutico del cancer. |
| CA2692050A1 (fr) * | 2007-06-12 | 2008-12-18 | F.Hoffmann-La Roche Ag | Thiazolopyrimidines et leur utilisation comme inhibiteurs de la phosphatidylinositol-3 kinase (pi3k) |
| CN101932587A (zh) * | 2007-09-24 | 2010-12-29 | 吉宁特有限公司 | 噻唑并嘧啶pi3k抑制剂化合物及使用方法 |
| CA2701292C (fr) * | 2007-10-25 | 2015-03-24 | Genentech, Inc. | Procede de preparation de composes de thienopyrimidine |
| GB0721095D0 (en) * | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
| US8536161B2 (en) | 2009-03-12 | 2013-09-17 | Genentech, Inc. | Combinations of phosphoinositide 3-kinase inhibitor compounds and chemotherapeutic agents for the treatment of hematopoietic malignancies |
| CA2772371A1 (fr) * | 2009-05-27 | 2010-12-02 | F. Hoffmann-La Roche Ag | Composes bicycliques indole-pyrimidine inhibiteurs de pi3k selectifs pour p110 delta et leurs procedes d'utilisation |
| CA2761445A1 (fr) | 2009-05-27 | 2010-12-02 | Genentech, Inc. | Composes pyrimidines bicycliques inhibiteurs de pi3k selectifs pour p110 delta, et procedes d'utilisation |
| AU2010314287A1 (en) * | 2009-10-12 | 2012-05-03 | F. Hoffmann-La Roche Ag | Combinations of a PI3K inhibitor and a MEK inhibitor |
| EP2558864A1 (fr) | 2010-04-16 | 2013-02-20 | Genentech, Inc. | Foxo3a utilisée comme biomarqueur prédictif pour l'efficacité d'un inhibiteur de la voie des kinases p13k/akt |
| US20140004209A1 (en) | 2010-12-22 | 2014-01-02 | Genentech, Inc. | Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms |
| RU2015140573A (ru) | 2013-02-25 | 2017-03-30 | Дженентек, Инк. | Способы и композиции для обнаружения и лечения устойчивого к лекарственным средствам мутанта акт |
-
0
- BE BE759493D patent/BE759493A/fr unknown
-
1970
- 1970-11-17 BG BG016080A patent/BG17799A3/xx unknown
- 1970-11-17 BG BG017732A patent/BG17800A3/xx unknown
- 1970-11-18 US US90841A patent/US3661908A/en not_active Expired - Lifetime
- 1970-11-23 CH CH1731270A patent/CH559210A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1514974A patent/CH568324A5/xx not_active IP Right Cessation
- 1970-11-23 CH CH1514674A patent/CH567029A5/xx not_active IP Right Cessation
- 1970-11-25 NL NL7017210A patent/NL7017210A/xx unknown
- 1970-11-25 DK DK601570AA patent/DK128781B/da unknown
- 1970-11-25 GB GB5614670A patent/GB1321316A/en not_active Expired
- 1970-11-25 NO NO04524/70A patent/NO129954B/no unknown
- 1970-11-26 IL IL35729A patent/IL35729A/xx unknown
- 1970-11-26 CA CA099166A patent/CA926865A/en not_active Expired
- 1970-11-26 SE SE7016054A patent/SE377938B/xx unknown
- 1970-11-26 IE IE1519/70A patent/IE34765B1/xx unknown
- 1970-11-26 FR FR7042531A patent/FR2073416B1/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| CH567029A5 (fr) | 1975-09-30 |
| IE34765B1 (en) | 1975-08-06 |
| CH568324A5 (fr) | 1975-10-31 |
| SE377938B (fr) | 1975-08-04 |
| IL35729A (en) | 1974-01-14 |
| FR2073416B1 (fr) | 1975-04-18 |
| US3661908A (en) | 1972-05-09 |
| DK128781B (da) | 1974-07-01 |
| GB1321316A (en) | 1973-06-27 |
| IE34765L (en) | 1971-05-26 |
| CA926865A (en) | 1973-05-22 |
| NO129954B (fr) | 1974-06-17 |
| BG17799A3 (bg) | 1973-12-25 |
| BG17800A3 (bg) | 1973-12-25 |
| CH559210A5 (fr) | 1975-02-28 |
| FR2073416A1 (fr) | 1971-10-01 |
| IL35729A0 (en) | 1971-01-28 |
| NL7017210A (fr) | 1971-05-28 |
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