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BG108440A - KRI''Al'An'Ihholin ... RICK, M ... 'O'ND FOR YOU ... GOVO'O PAL' -AVAN ... AND USED ... 'O M' FOR GOLF - ANAV ... OF L ... KAR''B ... BUT ... D'YOU - Google Patents

KRI''Al'An'Ihholin ... RICK, M ... 'O'ND FOR YOU ... GOVO'O PAL' -AVAN ... AND USED ... 'O M' FOR GOLF - ANAV ... OF L ... KAR''B ... BUT ... D'YOU

Info

Publication number
BG108440A
BG108440A BG108440A BG10844003A BG108440A BG 108440 A BG108440 A BG 108440A BG 108440 A BG108440 A BG 108440A BG 10844003 A BG10844003 A BG 10844003A BG 108440 A BG108440 A BG 108440A
Authority
BG
Bulgaria
Prior art keywords
ihholin
govo
anav
avan
kri
Prior art date
Application number
BG108440A
Other languages
Bulgarian (bg)
Other versions
BG66303B1 (en
Inventor
Ulrike Werthmann
Peter Sieger
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co.Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma Gmbh & Co.Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co.Kg
Publication of BG108440A publication Critical patent/BG108440A/en
Publication of BG66303B1 publication Critical patent/BG66303B1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pulmonology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)

Abstract

The invention relates to crystalline, water-free (1alpha, 2beta, 4beta, 5alpha, 7beta)-7-[(hydroxydi-2-thienylacetyl)oxy]-9,9-dimethyl-3-oxa-9-azo niatricyclo[3.3.1.02,4]nonane-bromide, to a method for its production, and to the use thereof in the production of a drug, especially in the production of an anticholinergic drug. 12 claims
BG108440A 2001-06-22 2003-12-12 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug BG66303B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10129710 2001-06-22
DE10215436 2002-04-08
PCT/EP2002/006291 WO2003000265A1 (en) 2001-06-22 2002-06-08 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug

Publications (2)

Publication Number Publication Date
BG108440A true BG108440A (en) 2004-08-31
BG66303B1 BG66303B1 (en) 2013-03-29

Family

ID=26009556

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108440A BG66303B1 (en) 2001-06-22 2003-12-12 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug

Country Status (37)

Country Link
EP (1) EP1401445B1 (en)
JP (1) JP2005504015A (en)
KR (2) KR101011353B1 (en)
CN (1) CN100586948C (en)
AR (1) AR037491A1 (en)
AT (1) ATE337006T1 (en)
AU (1) AU2002345016B2 (en)
BG (1) BG66303B1 (en)
BR (1) BR0210537A (en)
CA (1) CA2450961C (en)
CO (1) CO5550423A2 (en)
CY (1) CY1105223T1 (en)
CZ (1) CZ302786B6 (en)
DE (1) DE50207943D1 (en)
DK (1) DK1401445T3 (en)
EA (1) EA005813B1 (en)
EE (1) EE05316B1 (en)
EG (1) EG24851A (en)
ES (1) ES2271280T3 (en)
HR (1) HRP20031066B1 (en)
HU (1) HUP0400333A3 (en)
IL (2) IL159238A0 (en)
ME (1) ME00412B (en)
MX (1) MXPA03011718A (en)
MY (1) MY122779A (en)
NO (1) NO334301B1 (en)
NZ (1) NZ530690A (en)
PE (2) PE20030130A1 (en)
PL (1) PL208137B1 (en)
PT (1) PT1401445E (en)
RS (1) RS50441B (en)
SA (1) SA02230255B1 (en)
SI (1) SI1401445T1 (en)
SK (1) SK287262B6 (en)
TW (2) TWI261589B (en)
UY (1) UY27342A1 (en)
WO (1) WO2003000265A1 (en)

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ES2360963T3 (en) 2006-08-07 2011-06-10 Boehringer Ingelheim International Gmbh COMBINATIONS OF DRUGS FOR THE TREATMENT OF DISEASES OF THE RESPIRATORY ROUTES.
PE20080610A1 (en) 2006-08-22 2008-07-15 Boehringer Ingelheim Int NEW ENANTHOMERICALLY PURE BETA-AGONISTS, PROCEDURES FOR THEIR PREPARATION AND USE AS MEDICINES
GB0716026D0 (en) 2007-08-16 2007-09-26 Norton Healthcare Ltd An inhalable medicament
DK2215092T3 (en) 2007-10-19 2012-05-07 Boehringer Ingelheim Int Substituted piperidino dihydrothienopyrimidine
EP2093219A1 (en) 2008-02-22 2009-08-26 Boehringer Ingelheim International Gmbh Crystalline enantiomer free salt form of a betamimetic and its use as medicine
NZ592723A (en) 2008-12-19 2013-06-28 Boehringer Ingelheim Int Cyclic pyrimidin-4-carboxamides as ccr2 receptor antagonists for treatment of inflammation, asthma and copd
WO2010101538A2 (en) 2009-03-06 2010-09-10 Bilgic Mahmut New crystal forms
AP3170A (en) 2009-12-17 2015-03-31 Boehringer Ingelheim Int New CCR2 receptor antagonists and uses thereof
EP2513086B1 (en) 2009-12-17 2015-04-29 Boehringer Ingelheim International GmbH Novel antagonists for ccr2 and uses thereof
EP2528915B1 (en) 2010-01-29 2015-10-28 Boehringer Ingelheim International GmbH Substituted naphthyridines and their use as syk kinase inhibitors
EP2569295B1 (en) 2010-05-12 2014-11-19 Boehringer Ingelheim International GmbH New ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
EP2569298B1 (en) 2010-05-12 2015-11-25 Boehringer Ingelheim International GmbH Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
EP2571870B1 (en) 2010-05-17 2015-01-21 Boehringer Ingelheim International GmbH Ccr2 antagonists and uses thereof
US9018212B2 (en) 2010-05-25 2015-04-28 Boehringer Ingelheim International Gmbh Pyridazine carboxamides as CCR2 receptor antagonists
WO2011151251A1 (en) 2010-06-01 2011-12-08 Boehringer Ingelheim International Gmbh New ccr2 antagonists
TR201007108A2 (en) * 2010-08-25 2012-03-21 B�Lg�� Mahmut New tiotropium bromide crystal and production method.
WO2012101013A1 (en) 2011-01-28 2012-08-02 Boehringer Ingelheim International Gmbh Substituted pyridinyl-pyrimidines and their use as medicaments
TR201101897A2 (en) 2011-02-28 2012-09-21 Bi̇lgi̇ç Mahmut Crystal material containing tiotropium bromide
TR201102068A2 (en) 2011-03-03 2012-09-21 Bi̇lgi̇ç Mahmut Crystalline substances containing tiotropium bromide
TR201111589A2 (en) * 2011-03-03 2012-09-21 Bi̇lgi̇ç Mahmut Tiotropium bromide anhydrous crystal form.
EP2721025B1 (en) 2011-06-16 2015-11-25 Boehringer Ingelheim International Gmbh New selective ccr2 antagonists
WO2013010839A1 (en) 2011-07-15 2013-01-24 Boehringer Ingelheim International Gmbh Novel and selective ccr2 antagonists
AU2012288969B2 (en) 2011-07-26 2017-02-23 Boehringer Ingelheim International Gmbh Substituted quinolines and their use as medicaments
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
EP2782914B1 (en) 2011-11-25 2018-08-01 Adverio Pharma GmbH Method for producing substituted 5-fluoro-1h-pyrazolopyridines
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Also Published As

Publication number Publication date
PL364489A1 (en) 2004-12-13
AU2002345016B2 (en) 2008-04-17
SK287262B6 (en) 2010-04-07
EP1401445A1 (en) 2004-03-31
HRP20031066A2 (en) 2004-04-30
HUP0400333A3 (en) 2012-10-29
NZ530690A (en) 2005-05-27
DE50207943D1 (en) 2006-10-05
SK522004A3 (en) 2004-06-08
TWI261589B (en) 2006-09-11
MY122779A (en) 2006-05-31
PE20030130A1 (en) 2003-04-02
CZ302786B6 (en) 2011-11-09
EP1401445B1 (en) 2006-08-23
AR037491A1 (en) 2004-11-17
KR101011353B1 (en) 2011-01-28
CA2450961A1 (en) 2003-01-03
NO20035696D0 (en) 2003-12-19
EA200301293A1 (en) 2004-08-26
EE05316B1 (en) 2010-08-16
NO334301B1 (en) 2014-02-03
HRP20031066B1 (en) 2011-10-31
SA02230255B1 (en) 2006-10-31
UY27342A1 (en) 2003-02-28
RS50441B (en) 2010-03-02
EG24851A (en) 2010-10-27
IL159238A0 (en) 2004-06-01
KR100971616B1 (en) 2010-07-22
PT1401445E (en) 2006-10-31
BR0210537A (en) 2004-06-22
CA2450961C (en) 2010-03-30
CN1520294A (en) 2004-08-11
HK1068540A1 (en) 2005-04-29
PL208137B1 (en) 2011-03-31
ES2271280T3 (en) 2007-04-16
KR20040018285A (en) 2004-03-02
CN100586948C (en) 2010-02-03
ATE337006T1 (en) 2006-09-15
ME00412B (en) 2011-10-10
TW200617007A (en) 2006-06-01
YU99703A (en) 2006-05-25
SI1401445T1 (en) 2007-02-28
DK1401445T3 (en) 2006-11-27
PE20081305A1 (en) 2008-10-01
CY1105223T1 (en) 2010-03-03
MEP62008A (en) 2011-05-10
EA005813B1 (en) 2005-06-30
CZ2004120A3 (en) 2004-05-12
WO2003000265A1 (en) 2003-01-03
MXPA03011718A (en) 2004-12-06
CO5550423A2 (en) 2005-08-31
IL159238A (en) 2010-04-15
KR20090031638A (en) 2009-03-26
EE200400029A (en) 2004-04-15
BG66303B1 (en) 2013-03-29
JP2005504015A (en) 2005-02-10
HUP0400333A2 (en) 2004-12-28

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