CN110891575A - 治疗和/或预防光化性角化病的方法 - Google Patents
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- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
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| US201762469889P | 2017-03-10 | 2017-03-10 | |
| US62/469,889 | 2017-03-10 | ||
| PCT/US2018/021929 WO2018165647A1 (fr) | 2017-03-10 | 2018-03-12 | Méthodes de traitement et/ou de prévention de la kératose actinique |
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| EP (1) | EP3592355A4 (fr) |
| JP (3) | JP7502863B2 (fr) |
| KR (2) | KR20190141661A (fr) |
| CN (1) | CN110891575A (fr) |
| AU (2) | AU2018231144B2 (fr) |
| BR (1) | BR112019018687A2 (fr) |
| CA (1) | CA3055938A1 (fr) |
| IL (1) | IL269182B2 (fr) |
| MX (2) | MX387658B (fr) |
| TW (1) | TWI841523B (fr) |
| WO (1) | WO2018165647A1 (fr) |
| ZA (1) | ZA202100106B (fr) |
Cited By (1)
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| WO2025077886A1 (fr) * | 2023-10-13 | 2025-04-17 | 恩康药业科技(广州)有限公司 | Composé et procédé de traitement et/ou de prévention de la kératose actinique |
Families Citing this family (7)
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|---|---|---|---|---|
| US7968574B2 (en) * | 2004-12-28 | 2011-06-28 | Kinex Pharmaceuticals, Llc | Biaryl compositions and methods for modulating a kinase cascade |
| BR112019018687A2 (pt) * | 2017-03-10 | 2020-04-07 | Athenex Inc | métodos de tratamento e/ou prevenção da ceratose actínica |
| CN111278808B (zh) | 2017-09-07 | 2024-04-26 | 安兹克斯特殊目的有限责任公司 | 2-(5-(4-(2-吗啉代乙氧基)苯基)吡啶-2-基)-n-苄基乙酰胺的固体形式 |
| WO2019173533A1 (fr) * | 2018-03-07 | 2019-09-12 | Athenex HK Innovative Limited | Compositions et méthodes de traitement des troubles cutanés hyperprolifératifs |
| JP7296945B2 (ja) * | 2018-03-28 | 2023-06-23 | テルモ株式会社 | 医療デバイス |
| JP2022535267A (ja) * | 2019-06-05 | 2022-08-05 | アセネックス インコーポレイテッド | 乾癬を治療および/または予防する方法 |
| AU2022209830A1 (en) * | 2021-01-21 | 2023-08-03 | Sirnaomics, Inc. | Compositions and methods for treatment of skin cancers |
Citations (1)
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|---|---|---|---|---|
| US20110021555A1 (en) * | 2008-12-19 | 2011-01-27 | Graceway Pharmaceuticals, Llc | Lower dosage strength imiquimod formulations and shorter dosing regimens for treating actinic keratoses |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US7968574B2 (en) | 2004-12-28 | 2011-06-28 | Kinex Pharmaceuticals, Llc | Biaryl compositions and methods for modulating a kinase cascade |
| EP1836169B9 (fr) | 2004-12-28 | 2012-07-04 | Kinex Pharmaceuticals, LLC | Compositions et procédés de traitement de troubles impliquant une prolifération cellulaire |
| JP5564251B2 (ja) | 2006-06-29 | 2014-07-30 | キネックス ファーマシューティカルズ, エルエルシー | キナーゼカスケードを調節するためのビアリール組成物および方法 |
| US7538252B2 (en) * | 2006-09-05 | 2009-05-26 | Bipar Sciences, Inc. | Drug design for tubulin inhibitors, compositions, and methods of treatment thereof |
| US7939529B2 (en) | 2007-05-17 | 2011-05-10 | Kinex Pharmaceuticals, Llc | Process for the preparation of compositions for modulating a kinase cascade and methods of use thereof |
| TWI457336B (zh) | 2006-12-28 | 2014-10-21 | Kinex Pharmaceuticals Llc | 調節激酶級聯之組成物及方法 |
| US7935697B2 (en) | 2006-12-28 | 2011-05-03 | Kinex Pharmaceuticals, Llc | Compositions for modulating a kinase cascade and methods of use thereof |
| WO2008144045A1 (fr) | 2007-05-17 | 2008-11-27 | Kinex Pharmaceuticals, Llc | Procédé pour la préparation de compositions pour moduler une cascade de kinases et procédé d'utilisation de celui-ci |
| EP2143421A1 (fr) | 2008-07-07 | 2010-01-13 | Almirall Hermal GmbH | Composition topique pour le traitement de la kératose actinique |
| US8741857B1 (en) * | 2012-01-30 | 2014-06-03 | Lawrence Moy | Treatments for actinic keratoses |
| NZ606177A (en) * | 2012-01-30 | 2014-03-28 | Dolorgiet Gmbh & Co Kg | Compositions for the treatment of actinic keratosis |
| KR20150034209A (ko) | 2012-06-26 | 2015-04-02 | 델 마 파마슈티컬스 인코포레이티드 | 디안하이드로갈락티톨, 디아세틸디안하이드로갈락티톨, 디브로모둘시톨, 또는 그의 유사체 또는 유도체를 이용하여 유전학적 다형성이 있는 환자에 있어서 티로신-키나아제-억제제 내성 악성종양, ahi1 조절곤란 또는 돌연변이를 치료하는 방법 |
| BR112019018687A2 (pt) * | 2017-03-10 | 2020-04-07 | Athenex Inc | métodos de tratamento e/ou prevenção da ceratose actínica |
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- 2018-03-12 TW TW107108242A patent/TWI841523B/zh active
- 2018-03-12 KR KR1020197029678A patent/KR20190141661A/ko not_active Ceased
- 2018-03-12 WO PCT/US2018/021929 patent/WO2018165647A1/fr not_active Ceased
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- 2018-03-12 IL IL269182A patent/IL269182B2/en unknown
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- 2018-03-12 EP EP18764980.1A patent/EP3592355A4/fr active Pending
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- 2018-03-12 KR KR1020247017149A patent/KR20240090837A/ko active Pending
- 2018-03-12 JP JP2019549396A patent/JP7502863B2/ja active Active
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110021555A1 (en) * | 2008-12-19 | 2011-01-27 | Graceway Pharmaceuticals, Llc | Lower dosage strength imiquimod formulations and shorter dosing regimens for treating actinic keratoses |
Non-Patent Citations (2)
| Title |
|---|
| KINEX PHARMACEUTICALS: "Kinex Pharmaceuticals Announces Allowance of the Investigational New Drug (IND) application for KX2-391 Ointment by the United States Food and Drug Administration (FDA)", 《HTTPS://WWW.PRNEWSWIRE.COM/NEWS- RELEASES/KINEX-PHARMACEUTICALS-ANNOUNCES-ALLOWANCE-OF-THE-INVESTIGATIONAL-NEW-DRUG-IND-APPLICATION-FOR-KX2-391-OINTMENT-BY-THE-UNITED-STATES-FOOD-AND-DRUG-ADMINISTRATION-FDA-268466522.HTML》 * |
| 赵文丽: "FDA 接受 KX2-391 软膏治疗光化性角化病的研究性新药申请", 《国际药学研究杂志》 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2025077886A1 (fr) * | 2023-10-13 | 2025-04-17 | 恩康药业科技(广州)有限公司 | Composé et procédé de traitement et/ou de prévention de la kératose actinique |
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| MX2021013354A (es) | 2021-11-18 |
| US20180256589A1 (en) | 2018-09-13 |
| EP3592355A1 (fr) | 2020-01-15 |
| AU2018231144A1 (en) | 2019-10-03 |
| IL269182A (en) | 2019-11-28 |
| RU2019131757A3 (fr) | 2021-05-31 |
| BR112019018687A2 (pt) | 2020-04-07 |
| JP7502863B2 (ja) | 2024-06-19 |
| KR20240090837A (ko) | 2024-06-21 |
| US11497750B2 (en) | 2022-11-15 |
| WO2018165647A1 (fr) | 2018-09-13 |
| IL269182B2 (en) | 2023-11-01 |
| ZA202100106B (en) | 2022-08-31 |
| MX387658B (es) | 2025-03-18 |
| IL269182B1 (en) | 2023-07-01 |
| JP2020510042A (ja) | 2020-04-02 |
| US10617693B2 (en) | 2020-04-14 |
| KR20190141661A (ko) | 2019-12-24 |
| CA3055938A1 (fr) | 2018-09-13 |
| JP2025029010A (ja) | 2025-03-05 |
| US20230172942A1 (en) | 2023-06-08 |
| RU2019131757A (ru) | 2021-04-12 |
| EP3592355A4 (fr) | 2021-01-06 |
| AU2024201828A1 (en) | 2024-05-02 |
| US20200197405A1 (en) | 2020-06-25 |
| TW201842913A (zh) | 2018-12-16 |
| TWI841523B (zh) | 2024-05-11 |
| MX2019010707A (es) | 2020-01-15 |
| AU2018231144B2 (en) | 2023-12-21 |
| JP2023015269A (ja) | 2023-01-31 |
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