ES2366278T3 - Formulación de liberación controlada (albuterol). - Google Patents

Formulación de liberación controlada (albuterol). Download PDF

Info

Publication number: ES2366278T3
Authority: ES; Spain
Prior art keywords: dosage form; controlled release; release dosage; solid controlled; patient
Prior art date: 1995-11-03
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

ES96940352T

Other languages

English (en)

Spanish (es)

Inventor

Anand R. Baichwal

Troy W. Mccall

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Penwest Pharmaceuticals Co

Original Assignee

Penwest Pharmaceuticals Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-11-03

Filing date

1996-11-04

Publication date

2011-10-18

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24207743&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES2366278(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1996-11-04 Application filed by Penwest Pharmaceuticals Co filed Critical Penwest Pharmaceuticals Co

2011-10-18 Application granted granted Critical

2011-10-18 Publication of ES2366278T3 publication Critical patent/ES2366278T3/es

2016-11-04 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Links

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239000000344 soap Substances 0.000 description 1
235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
229940080313 sodium starch Drugs 0.000 description 1
239000003381 stabilizer Substances 0.000 description 1
150000003431 steroids Chemical class 0.000 description 1
239000000021 stimulant Substances 0.000 description 1
KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 description 1
150000008163 sugars Chemical class 0.000 description 1
229960000894 sulindac Drugs 0.000 description 1
MLKXDPUZXIRXEP-MFOYZWKCSA-N sulindac Chemical compound CC1=C(CC(O)=O)C2=CC(F)=CC=C2\C1=C/C1=CC=C(S(C)=O)C=C1 MLKXDPUZXIRXEP-MFOYZWKCSA-N 0.000 description 1
230000008961 swelling Effects 0.000 description 1
230000001975 sympathomimetic effect Effects 0.000 description 1
229940064707 sympathomimetics Drugs 0.000 description 1
208000024891 symptom Diseases 0.000 description 1
239000011885 synergistic combination Substances 0.000 description 1
229920002994 synthetic fiber Polymers 0.000 description 1
239000002278 tabletting lubricant Substances 0.000 description 1
229960000195 terbutaline Drugs 0.000 description 1
KFVSLSTULZVNPG-UHFFFAOYSA-N terbutaline sulfate Chemical compound [O-]S([O-])(=O)=O.CC(C)(C)[NH2+]CC(O)C1=CC(O)=CC(O)=C1.CC(C)(C)[NH2+]CC(O)C1=CC(O)=CC(O)=C1 KFVSLSTULZVNPG-UHFFFAOYSA-N 0.000 description 1
229960005105 terbutaline sulfate Drugs 0.000 description 1
229960002180 tetracycline Drugs 0.000 description 1
229930101283 tetracycline Natural products 0.000 description 1
235000019364 tetracycline Nutrition 0.000 description 1
150000003522 tetracyclines Chemical class 0.000 description 1
BJORNXNYWNIWEY-UHFFFAOYSA-N tetrahydrozoline hydrochloride Chemical compound Cl.N1CCN=C1C1C2=CC=CC=C2CCC1 BJORNXNYWNIWEY-UHFFFAOYSA-N 0.000 description 1
229940021790 tetrahydrozoline hydrochloride Drugs 0.000 description 1
229960000278 theophylline Drugs 0.000 description 1
239000004408 titanium dioxide Substances 0.000 description 1
238000012546 transfer Methods 0.000 description 1
229960005294 triamcinolone Drugs 0.000 description 1
GFNANZIMVAIWHM-OBYCQNJPSA-N triamcinolone Chemical compound O=C1C=C[C@]2(C)[C@@]3(F)[C@@H](O)C[C@](C)([C@@]([C@H](O)C4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 GFNANZIMVAIWHM-OBYCQNJPSA-N 0.000 description 1
125000005591 trimellitate group Chemical group 0.000 description 1
229940124549 vasodilator Drugs 0.000 description 1
239000003071 vasodilator agent Substances 0.000 description 1
239000003981 vehicle Substances 0.000 description 1
125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
229940088594 vitamin Drugs 0.000 description 1
239000011782 vitamin Substances 0.000 description 1
229930003231 vitamin Natural products 0.000 description 1
235000013343 vitamin Nutrition 0.000 description 1
230000004580 weight loss Effects 0.000 description 1
239000000080 wetting agent Substances 0.000 description 1
229960001095 xylometazoline hydrochloride Drugs 0.000 description 1
UHVMMEOXYDMDKI-JKYCWFKZSA-L zinc;1-(5-cyanopyridin-2-yl)-3-[(1s,2s)-2-(6-fluoro-2-hydroxy-3-propanoylphenyl)cyclopropyl]urea;diacetate Chemical compound [Zn+2].CC([O-])=O.CC([O-])=O.CCC(=O)C1=CC=C(F)C([C@H]2[C@H](C2)NC(=O)NC=2N=CC(=CC=2)C#N)=C1O UHVMMEOXYDMDKI-JKYCWFKZSA-L 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08J—WORKING-UP; GENERAL PROCESSES OF COMPOUNDING; AFTER-TREATMENT NOT COVERED BY SUBCLASSES C08B, C08C, C08F, C08G or C08H
- C08J3/00—Processes of treating or compounding macromolecular substances
- C08J3/02—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques
- C08J3/03—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques in aqueous media
- C08J3/075—Macromolecular gels

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Dispersion Chemistry (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Emergency Medicine (AREA)
Inorganic Chemistry (AREA)
Polymers & Plastics (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Pulmonology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

ES96940352T 1995-11-03 1996-11-04 Formulación de liberación controlada (albuterol). Expired - Lifetime ES2366278T3 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US553008		1983-11-17
US08/553,008 US5662933A (en)	1993-09-09	1995-11-03	Controlled release formulation (albuterol)

Publications (1)

Publication Number	Publication Date
ES2366278T3 true ES2366278T3 (es)	2011-10-18

Family

ID=24207743

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ES96940352T Expired - Lifetime ES2366278T3 (es)	1995-11-03	1996-11-04	Formulación de liberación controlada (albuterol).

Country Status (12)

Country	Link
US (2)	US5662933A (fr)
EP (2)	EP2286796A3 (fr)
JP (1)	JP3250737B2 (fr)
KR (2)	KR100264024B1 (fr)
AT (1)	ATE507820T1 (fr)
AU (1)	AU7725396A (fr)
CA (1)	CA2208230C (fr)
DE (1)	DE69638364D1 (fr)
DK (1)	DK0804166T3 (fr)
ES (1)	ES2366278T3 (fr)
MX (1)	MX9704910A (fr)
WO (1)	WO1997016172A1 (fr)

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1995
- 1995-11-03 US US08/553,008 patent/US5662933A/en not_active Expired - Lifetime
1996
- 1996-11-04 EP EP10178632A patent/EP2286796A3/fr not_active Withdrawn
- 1996-11-04 AT AT96940352T patent/ATE507820T1/de active
- 1996-11-04 DK DK96940352.6T patent/DK0804166T3/da active
- 1996-11-04 ES ES96940352T patent/ES2366278T3/es not_active Expired - Lifetime
- 1996-11-04 DE DE69638364T patent/DE69638364D1/de not_active Expired - Lifetime
- 1996-11-04 KR KR1019970704570A patent/KR100264024B1/ko not_active Expired - Fee Related
- 1996-11-04 JP JP51763797A patent/JP3250737B2/ja not_active Expired - Fee Related
- 1996-11-04 EP EP96940352A patent/EP0804166B1/fr not_active Expired - Lifetime
- 1996-11-04 WO PCT/US1996/017991 patent/WO1997016172A1/fr active IP Right Grant
- 1996-11-04 AU AU77253/96A patent/AU7725396A/en not_active Abandoned
- 1996-11-04 CA CA002208230A patent/CA2208230C/fr not_active Expired - Fee Related
1997
- 1997-06-27 MX MX9704910A patent/MX9704910A/es active IP Right Grant
- 1997-07-01 US US08/886,496 patent/US5958456A/en not_active Expired - Lifetime
2000
- 2000-01-07 KR KR1020000000749A patent/KR20000018064A/ko not_active Ceased

Also Published As

Publication number	Publication date
JPH10507210A (ja)	1998-07-14
EP2286796A3 (fr)	2012-02-22
AU7725396A (en)	1997-05-22
KR20000018064A (ko)	2000-04-06
MX9704910A (es)	1998-06-30
DE69638364D1 (de)	2011-06-16
JP3250737B2 (ja)	2002-01-28
DK0804166T3 (da)	2011-08-15
EP0804166A1 (fr)	1997-11-05
EP0804166A4 (fr)	2004-12-29
US5662933A (en)	1997-09-02
WO1997016172A1 (fr)	1997-05-09
EP2286796A2 (fr)	2011-02-23
ATE507820T1 (de)	2011-05-15
US5958456A (en)	1999-09-28
CA2208230C (fr)	2001-12-25
EP0804166B1 (fr)	2011-05-04
CA2208230A1 (fr)	1997-05-09
KR100264024B1 (ko)	2000-09-01

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