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FI891021A0 - Menetelmä lääkeaineina käyttökelpoisten 1,2,4-triatsolijohdannaisten valmistamiseksi - Google Patents

Menetelmä lääkeaineina käyttökelpoisten 1,2,4-triatsolijohdannaisten valmistamiseksi

Info

Publication number
FI891021A0
FI891021A0 FI891021A FI891021A FI891021A0 FI 891021 A0 FI891021 A0 FI 891021A0 FI 891021 A FI891021 A FI 891021A FI 891021 A FI891021 A FI 891021A FI 891021 A0 FI891021 A0 FI 891021A0
Authority
FI
Finland
Prior art keywords
drug
preparation
triazole derivatives
derivatives useful
triazole
Prior art date
Application number
FI891021A
Other languages
English (en)
Swedish (sv)
Other versions
FI97382C (fi
FI891021A7 (fi
FI97382B (fi
Inventor
Sadao Oida
Yawara Tajima
Toshiyuki Konosu
Masayuki Iwata
Noriko Takeda
Takeo Miyaoka
Hideo Takeshiba
Toshiro Nakanishi
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of FI891021A0 publication Critical patent/FI891021A0/fi
Publication of FI891021A7 publication Critical patent/FI891021A7/fi
Application granted granted Critical
Publication of FI97382B publication Critical patent/FI97382B/fi
Publication of FI97382C publication Critical patent/FI97382C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647Triazoles; Hydrogenated triazoles
    • A01N43/6531,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24Halogenated aromatic hydrocarbons with unsaturated side chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46Friedel-Crafts reactions
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/82Ketones containing a keto group bound to a six-membered aromatic ring containing hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI891021A 1988-03-04 1989-03-03 Menetelmä lääkeaineina käyttökelpoisten 1,2,4-triatsolijohdannaisten valmistamiseksi FI97382C (fi)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
JP5131288 1988-03-04
JP5131288 1988-03-04
JP6868188 1988-03-23
JP6868188 1988-03-23
JP25015888 1988-10-04
JP25015888 1988-10-04
JP26121188 1988-10-17
JP26121188 1988-10-17

Publications (4)

Publication Number Publication Date
FI891021A0 true FI891021A0 (fi) 1989-03-03
FI891021A7 FI891021A7 (fi) 1989-09-05
FI97382B FI97382B (fi) 1996-08-30
FI97382C FI97382C (fi) 1996-12-10

Family

ID=27462619

Family Applications (1)

Application Number Title Priority Date Filing Date
FI891021A FI97382C (fi) 1988-03-04 1989-03-03 Menetelmä lääkeaineina käyttökelpoisten 1,2,4-triatsolijohdannaisten valmistamiseksi

Country Status (11)

Country Link
EP (1) EP0332387B1 (fi)
KR (1) KR890014500A (fi)
AU (1) AU622639B2 (fi)
DE (1) DE68910853T2 (fi)
DK (1) DK105189A (fi)
ES (1) ES2061975T3 (fi)
FI (1) FI97382C (fi)
HU (1) HUT53889A (fi)
IE (1) IE64189B1 (fi)
NO (1) NO171272C (fi)
NZ (1) NZ228236A (fi)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
US5206364A (en) * 1988-08-13 1993-04-27 Pfizer Inc. Triazole antifungal agents
IE903395A1 (en) * 1989-09-26 1991-04-10 Takeda Chemical Industries Ltd Triazole compounds, their production and use
TW206224B (fi) * 1989-12-14 1993-05-21 Takeda Pharm Industry Co Ltd
CA2031892C (en) * 1989-12-25 2000-08-01 Minoru Tokizawa Triazole derivatives
US5278175A (en) * 1990-02-02 1994-01-11 Pfizer Inc. Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
EP0446877A3 (en) * 1990-03-15 1992-05-06 Takeda Chemical Industries, Ltd. Triazoles, their production and use
IT1240676B (it) * 1990-04-24 1993-12-17 Agrimont Spa Composizioni ad attivita' erbicida
ES2024332A6 (es) * 1990-10-08 1992-02-16 Uriach & Cia Sa J Procedimiento para la obtencion de nuevas sulfonamidas.
AU1762492A (en) * 1991-03-27 1992-11-02 Schering Corporation Preparation of chiral hydroxyketones
WO1992017433A1 (en) * 1991-03-27 1992-10-15 Schering Corporation Preparation of chiral hydroxyketones
EP0510700A3 (en) * 1991-04-26 1992-12-16 Takeda Chemical Industries, Ltd. Azole compounds, their production and use
ES2038906B1 (es) * 1991-09-04 1994-02-16 Uriach & Cia Sa J Procedimiento para la obtencion de nuevas oxazoilidinas.
GB9121456D0 (en) * 1991-10-10 1991-11-27 Pfizer Ltd Triazole antifungal agents
US5426233A (en) * 1992-03-25 1995-06-20 Schering Corporation Preparation of chiral hydroxyketones
TW218017B (fi) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
ES2051226B1 (es) * 1992-07-15 1994-12-16 Uriach & Cia Sa J Procedimiento para la obtencion del (-)-(2r,3r)-2-(2,4-diclorofenil)-3-(n-metanosulfonil-n-metilamino)-1-(1h-1,2,4-triazol-1-il)-2-butanol.
ES2099004B1 (es) * 1993-02-11 1998-01-16 Uriach & Cia Sa J Nuevos antifungicos activos por via oral.
ES2062941B1 (es) * 1993-03-15 1995-10-01 Uriach & Cia Sa J Nuevos derivados de azol activos por via oral.
TW297813B (fi) * 1993-09-24 1997-02-11 Takeda Pharm Industry Co Ltd
US5349099A (en) * 1993-12-13 1994-09-20 Schering Corporation Process for preparing intermediates for the synthesis of antifungal agents
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
CA2145458A1 (en) * 1994-03-28 1995-09-29 Hiroki Kodama Triazole compound and production process and use thereof
AU2630795A (en) * 1994-06-10 1996-01-05 Tokyo Tanabe Company Limited Triazole compound and antifungal agent containing the same as active ingredient
TW318841B (fi) 1995-02-17 1997-11-01 Takeda Pharm Industry Co Ltd
DK0841327T3 (da) * 1995-04-06 2002-01-21 Sankyo Co Triazolantisvampemiddel
CA2180091A1 (en) * 1995-07-08 1997-01-09 Hiroki Kodama Optically active triazole derivative, process for producing the same, antifungal agent, and method for using the same
KR970705560A (ko) * 1995-08-02 1997-10-09 호아껭 우리아치 토렐로 항진균 활성을 갖는 신규한 카르복사미드(new carboxamides with antifungal activity)
ES2112774B1 (es) * 1995-10-20 1999-05-16 Uriach & Cia Sa J Nuevos derivados azolicos con actividad antifungica.
US6133485A (en) * 1998-04-15 2000-10-17 Synphar Laboratories, Inc. Asymmetric synthesis of 2-(2,4-difluorophenyl)-1-heterocycl-1-yl butan-2,3-diols
GB9924692D0 (en) 1999-10-20 1999-12-22 Hoechst Schering Agrevo Gmbh Wood treatment
AU2007201000B2 (en) * 2000-09-05 2008-07-03 Donaldson Company, Inc. Polymer fine fiber and fine fiber layer
CN1819998B (zh) * 2003-07-18 2010-09-08 株式会社钟化 光学活性卤代醇衍生物及用其的光学活性环氧醇衍生物的制法
MX2008013305A (es) * 2006-04-20 2008-10-27 Du Pont Agentes heterociclicos de cinco miembros para el control de plagas de invertebrados.
WO2019216810A1 (en) * 2018-05-07 2019-11-14 Constantin Urban New antifungal compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4654332A (en) * 1979-03-07 1987-03-31 Imperial Chemical Industries Plc Heterocyclic compounds
US4482558A (en) * 1982-06-18 1984-11-13 Pfizer Inc. Antifungal amide and urea derivatives of (3-amino-2-aryl-2-hydroxyprop-1-yl)-1H-1,2,4-triazoles
DE3307218A1 (de) * 1983-03-02 1984-09-06 Bayer Ag, 5090 Leverkusen Substituierte diazolylalkyl-carbinole, verfahren zu ihrer herstellung und ihre verwendung als antimykotische mittel
CH658654A5 (de) * 1983-03-04 1986-11-28 Sandoz Ag Azolderivate, verfahren zu ihrer herstellung und mittel die diese verbindungen enthalten.
GB8306351D0 (en) * 1983-03-08 1983-04-13 Ici Plc Azole fungicides
US4483863A (en) * 1984-01-20 1984-11-20 Pfizer Inc. Triazole antifungal agents
GB8412750D0 (en) * 1984-05-18 1984-06-27 Ici Plc Heterocyclic compounds
DE3530799A1 (de) * 1985-08-29 1987-03-05 Hoechst Ag Azolyl-cyclopropyl-ethanol-derivate, verfahren zu ihrer herstellung und ihre verwendung
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
HUT53889A (en) 1990-12-28
AU622639B2 (en) 1992-04-16
IE890712L (en) 1989-09-04
NO171272C (no) 1993-02-17
EP0332387B1 (en) 1993-11-24
AU3105189A (en) 1989-09-07
DK105189D0 (da) 1989-03-03
EP0332387A1 (en) 1989-09-13
NZ228236A (en) 1991-02-26
NO890926D0 (no) 1989-03-03
FI97382C (fi) 1996-12-10
KR890014500A (ko) 1989-10-24
FI891021A7 (fi) 1989-09-05
IE64189B1 (en) 1995-07-12
NO890926L (no) 1989-09-05
DE68910853T2 (de) 1994-06-30
DE68910853D1 (de) 1994-01-05
DK105189A (da) 1989-09-05
ES2061975T3 (es) 1994-12-16
FI97382B (fi) 1996-08-30
NO171272B (no) 1992-11-09

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Legal Events

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BB Publication of examined application
MM Patent lapsed
MM Patent lapsed

Owner name: SANKYO COMPANY LIMITED