[go: up one dir, main page]

HK1049836A1 - 新的偶合方法 - Google Patents

新的偶合方法 Download PDF

Info

Publication number
HK1049836A1
HK1049836A1 HK03101949.7A HK03101949A HK1049836A1 HK 1049836 A1 HK1049836 A1 HK 1049836A1 HK 03101949 A HK03101949 A HK 03101949A HK 1049836 A1 HK1049836 A1 HK 1049836A1
Authority
HK
Hong Kong
Prior art keywords
coupling process
new coupling
compound
formula
new
Prior art date
Application number
HK03101949.7A
Other languages
English (en)
Inventor
Alvhall Jorgen
Edvardsson Daniel
Ioannidis Panagiotis
Sjogren Magnus
Szonyi Maria
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HK1049836A1 publication Critical patent/HK1049836A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
HK03101949.7A 2000-02-07 2001-01-30 新的偶合方法 HK1049836A1 (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0000382 2000-02-07
SE0000382A SE0000382D0 (sv) 2000-02-07 2000-02-07 New process
PCT/SE2001/000177 WO2001056986A1 (en) 2000-02-07 2001-01-30 New coupling process

Publications (1)

Publication Number Publication Date
HK1049836A1 true HK1049836A1 (zh) 2003-05-30

Family

ID=20278363

Family Applications (1)

Application Number Title Priority Date Filing Date
HK03101949.7A HK1049836A1 (zh) 2000-02-07 2001-01-30 新的偶合方法

Country Status (20)

Country Link
US (1) US6518434B2 (zh)
EP (1) EP1257533A1 (zh)
JP (1) JP2003521534A (zh)
KR (1) KR20020073202A (zh)
CN (1) CN1227227C (zh)
AU (1) AU769009B2 (zh)
BR (1) BR0108130A (zh)
CA (1) CA2396743A1 (zh)
CZ (1) CZ20022675A3 (zh)
HK (1) HK1049836A1 (zh)
HU (1) HUP0300381A3 (zh)
IL (1) IL150573A0 (zh)
MX (1) MXPA02007388A (zh)
NO (1) NO20023714L (zh)
NZ (1) NZ519946A (zh)
PL (1) PL358006A1 (zh)
SE (1) SE0000382D0 (zh)
SK (1) SK11252002A3 (zh)
WO (1) WO2001056986A1 (zh)
ZA (1) ZA200205235B (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR036187A1 (es) * 2001-07-24 2004-08-18 Adir Un proceso para la preparacion de perindopril, compuestos analogos y sus sales, compuesto intermediario 2,5-dioxo-oxazolidina y proceso para preparar un intermediario
CN104628586A (zh) * 2005-09-29 2015-05-20 中化帝斯曼制药有限公司荷兰公司 用于酯化有机酸的方法
WO2010059420A1 (en) * 2008-11-18 2010-05-27 Invista Technologies S.A.R.L. 1,2-diaminocyclohexane and chemical process

Family Cites Families (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH365385A (de) 1958-01-13 1962-11-15 Geigy Ag J R Verfahren zur Herstellung von a-substituierten Glycinen bzw. Glycinestern
GB1153792A (en) 1965-10-12 1969-05-29 Pfizer & Co C Pharmaceutical Compositions
SE372006B (zh) 1971-09-13 1974-12-09 Haessle Ab
US3784562A (en) 1972-06-21 1974-01-08 Squibb & Sons Inc Methyl acetoacetic ester enamine of d-2-(1,4-cyclohexadien-1-yl)glycine, sodium salt-dimethylformamide adduct
DE2807286A1 (de) 1978-02-21 1979-08-23 Bayer Ag Stereoselektive spaltung von phenylglycinderivaten und 4-hydroxyphenylglycinderivaten mit enzymharzen
DE3003653A1 (de) 1980-02-01 1981-08-06 Hoechst Ag, 6000 Frankfurt Verfahren zur herstellung von n-substituierten oxazolindionen-(2,4)
US4686295A (en) 1982-03-10 1987-08-11 Usv Pharmaceutical Corporation N-carboxy anhydride intermediates
DE3227055A1 (de) 1982-07-20 1984-01-26 Hoechst Ag, 6230 Frankfurt Neue derivate der 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure als zwischenstufe und verfahren zu deren herstellung
DE3303344A1 (de) 1983-02-02 1984-08-02 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von n-alkylierten aminosaeuren und deren estern
FR2555577B1 (fr) * 1983-11-24 1987-07-31 Flork Michel Nouveaux derives de peptides, leur procede de preparation et leur emploi comme reactif biologique
EP0174358A1 (en) 1984-03-01 1986-03-19 ALKALOIDA VEGYéSZETI GYáR Novel diastereomer salts of phenylalanine and n-acyl derivatives thereof and process for the separation of optically active phenylalanine and n-acyl derivatives thereof
GB8408801D0 (en) 1984-04-05 1984-05-16 Bp Chem Int Ltd Process for making esters
EP0168769A3 (en) * 1984-07-16 1989-02-08 Merck & Co. Inc. Process for preparing carboxyalkyl dipeptides
DE3623397A1 (de) 1986-07-11 1988-01-14 Boehringer Mannheim Gmbh Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
GB8631020D0 (en) 1986-12-30 1987-02-04 Janssen Pharmaceutica Nv 1-methyl-1h-imidazole-5-carboxylic acid derivatives
JPS6445350A (en) 1987-08-13 1989-02-17 Sagami Chem Res Production of n-substituted-l-amino acid derivative
US5028693A (en) 1988-03-11 1991-07-02 Bioresearch, Inc. Urethane-protected amino acid-N-carboxyanhydrides
US4946942A (en) 1988-03-11 1990-08-07 Bioresearch, Inc. Urethane-protected amino acid-N-carboxyanhydrides
JPH01254651A (ja) * 1988-04-04 1989-10-11 Kanegafuchi Chem Ind Co Ltd Ｎ↑２−（１−カルボキシ−３−フエニルプロピル）−ｌ−リジン誘導体及び該化合物を用いるリジノプリルの製造法
US4935328A (en) * 1988-04-07 1990-06-19 E. I. Du Pont De Nemours And Company Monofunctional amines as adjuvant for liquid electrostatic developers
DE4011171A1 (de) 1990-04-06 1991-10-10 Degussa Herstellung von (alpha)-aminosaeure-2,2,2,-trifluorethylester
US5892112A (en) 1990-11-21 1999-04-06 Glycomed Incorporated Process for preparing synthetic matrix metalloprotease inhibitors
CA2056911C (en) 1990-12-11 1998-09-22 Yuuichi Nagano Hiv protease inhibitors
AU653060B2 (en) 1991-08-23 1994-09-15 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivative and platelet agglutination inhibitor
US5650508A (en) 1991-12-27 1997-07-22 Georgia Tech Research Corporation Peptide ketoamides
GB9201755D0 (en) 1992-01-28 1992-03-11 British Bio Technology Compounds
TW223629B (zh) 1992-03-06 1994-05-11 Hoffmann La Roche
GB9206757D0 (en) 1992-03-27 1992-05-13 Ferring Bv Novel peptide receptor ligands
SI9200213A (en) * 1992-09-16 1994-03-31 Krka Process for preparing alkyl-l-alanil-l-proline derivates
SK37595A3 (en) 1992-09-25 1995-07-11 Bio Mega Boehringer Ingelheim N-(hydroxyethyl) butanediamine derivatives as renim inhibitors
ZA951617B (en) 1994-03-04 1997-02-27 Lilly Co Eli Antithrombotic agents.
FR2725991B1 (fr) 1994-10-24 1997-01-17 Univ Montpellier Ii Procede de synthese peptidique a partir des n-(n'-(r')-n' -nitrosocarbamoyls) aminoacides
US5994583A (en) 1996-05-22 1999-11-30 The Scripps Research Institute Two step synthesis of D- and L- α-amino acids and D- and L- α-amino-aldehydes
EP0922030A1 (en) 1996-08-23 1999-06-16 Pfizer Inc. Arylsulfonylamino hydroxamic acid derivatives
AR013084A1 (es) 1997-06-19 2000-12-13 Astrazeneca Ab Derivados de amidino utiles como inhibidores de la trombina, composicion farmaceutica, utilizacion de dichos compuestos para la preparacion demedicamentos y proceso para la preparacion de los compuestos mencionados
DE19920907A1 (de) 1999-05-06 2000-11-09 Basf Ag Verfahren zur Herstellung eines Cyclohexylglycin-Bausteins

Also Published As

Publication number Publication date
BR0108130A (pt) 2003-02-25
HUP0300381A3 (en) 2005-06-28
PL358006A1 (en) 2004-08-09
NO20023714D0 (no) 2002-08-06
US6518434B2 (en) 2003-02-11
SE0000382D0 (sv) 2000-02-07
WO2001056986A1 (en) 2001-08-09
NO20023714L (no) 2002-10-03
KR20020073202A (ko) 2002-09-19
CZ20022675A3 (cs) 2002-11-13
IL150573A0 (en) 2003-02-12
ZA200205235B (en) 2003-09-29
MXPA02007388A (es) 2002-12-09
SK11252002A3 (sk) 2003-02-04
US20020128452A1 (en) 2002-09-12
AU3251601A (en) 2001-08-14
JP2003521534A (ja) 2003-07-15
HUP0300381A2 (hu) 2003-06-28
CN1227227C (zh) 2005-11-16
AU769009B2 (en) 2004-01-15
CA2396743A1 (en) 2001-08-09
EP1257533A1 (en) 2002-11-20
CN1398255A (zh) 2003-02-19
NZ519946A (en) 2004-11-26

Similar Documents

Publication Publication Date Title
WO2002083662A3 (en) Azo compounds and process of producing the same and novel intermediate compounds used in the process of producing azo compounds
WO2002032898A3 (de) Neue anticholinergika, verfahren zu deren herstellung und deren verwendung als arzneimittel
AU2003277795A1 (en) A method of production of (-)-(s)-3-(1-(dimethylamino)ethyl)phenyl-n-ethyl-n-methylcarbamate
EP1156042A4 (en) PROCESS FOR THE PREPARATION OF GLYCEROL CARBONATE
WO2003014110A1 (fr) Derive de benzazepine, son procede de preparation et d'utilisation
CA2309474A1 (en) New 4-arylpiperidine derivatives for the treatment of pruritus
AP2001002194A0 (en) Novel process for the preparation of pyrazolopyrimidinones.
WO2002044161A3 (en) A process for the preparation of taxan derivatives
HK1049836A1 (zh) 新的偶合方法
IL145449A0 (en) Processes for preparing pesticidal intermediates
AU2002365378A1 (en) Process for preparing 3,3',6,6'-tetraalkyl-2,2'-biphenols and 3,3',6,6'-tetraalkyl-5,5'-dihalo-2,2'-biphenols
GB0019124D0 (en) Novel process
MXPA02001406A (es) Heterociclilos-2h-cromenos substituidos.
AU8459401A (en) Process for preparing a substituted imidazopyridine compound
EP1199312A3 (en) Process for producing an amide compound
HK1052350A1 (zh) 一種合成嗎啉基苯類化合物的新方法
CA2276310A1 (en) Process for the production of tetrazolylbenzopyrans
SE0101323D0 (sv) New process
AP2001002195A0 (en) Novel process for the preparation of pyrazolopyrimidinones.
IN2012DN02301A (zh)
AU2003226448A1 (en) Production method of 2,6-dihalopurine
WO2001010862A3 (de) Substituierte heterocyclylbenzofurane
EP1253144A4 (en) 1,3,4-OXADIAZOLE DERIVATIVES AND A METHOD FOR THE PRODUCTION THEREOF
CA2390934A1 (en) Process for producing benzylamine compound
EP1253143A4 (en) 1,3,4-OXADIAZOLE DERIVATIVES AND A METHOD FOR THE PRODUCTION THEREOF