HUP1100453A2 - Carboxamides with sterane skeleton as h3 antagonists - Google Patents

Carboxamides with sterane skeleton as h3 antagonists

Info

Publication number: HUP1100453A2
Authority: HU; Hungary
Prior art keywords: carboxamides; antagonists; sterane; skeleton; sterane skeleton
Prior art date: 2011-08-19

Application number

HU1100453A

Other languages

Hungarian (hu)

Inventor

Istvan Dr Ledneczki

Sandor Maho

Eszter Gabor

Pal Dr Tapolcsanyi

Bela Kiss

Ottilia Dr Balazs

Eva Dr Schmidt

Original Assignee

Richter Gedeon Nyrt

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-08-19

Filing date

2011-08-19

Publication date

2013-02-28

2011-08-19 Application filed by Richter Gedeon Nyrt filed Critical Richter Gedeon Nyrt

2011-08-19 Priority to HU1100453A priority Critical patent/HUP1100453A2/en

2012-08-17 Priority to PCT/HU2012/000075 priority patent/WO2013027073A1/en

2013-02-28 Publication of HUP1100453A2 publication Critical patent/HUP1100453A2/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0055—Estrane derivatives not substituted in position 17
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0077—Ethers

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

HU1100453A 2011-08-19 2011-08-19 Carboxamides with sterane skeleton as h3 antagonists HUP1100453A2 (en)

Priority Applications (2)

Application Number	Priority Date	Filing Date	Title
HU1100453A HUP1100453A2 (en)	2011-08-19	2011-08-19	Carboxamides with sterane skeleton as h3 antagonists
PCT/HU2012/000075 WO2013027073A1 (en)	2011-08-19	2012-08-17	Histamine h3 antagonist steroidal carboxamides

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
HU1100453A HUP1100453A2 (en)	2011-08-19	2011-08-19	Carboxamides with sterane skeleton as h3 antagonists

Publications (1)

Publication Number	Publication Date
HUP1100453A2 true HUP1100453A2 (en)	2013-02-28

Family

ID=89990402

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU1100453A HUP1100453A2 (en)	2011-08-19	2011-08-19	Carboxamides with sterane skeleton as h3 antagonists

Country Status (2)

Country	Link
HU (1)	HUP1100453A2 (en)
WO (1)	WO2013027073A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2022113008A1 (en)	2020-11-27	2022-06-02	Richter Gedeon Nyrt.	Histamine h3 receptor antagonists/inverse agonists for the treatment of autism spectrum disorder

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1338308A (en) *	1961-08-11	1963-09-27	Roussel Uclaf	Aromatic steroids substituted in position 3 and method of preparation
AU2002243643A1 (en) *	2001-01-25	2002-08-06	Yale University	Estradiol-16alpha-carboxylic acid esters as locally active estrogens
WO2004085345A2 (en) *	2003-03-21	2004-10-07	Yale University	15α-SUBSTITUTED ESTRADIOL CARBOXYLIC ACID ESTERS AS LOCALLY ACTIVE ESTROGENS
GB0306718D0 (en) *	2003-03-24	2003-04-30	Sterix Ltd	Compound
US7687486B2 (en) *	2003-04-29	2010-03-30	Florida Agricultural & Mechanical University	Selective estrogen receptor modulators
US7345034B2 (en)	2004-04-07	2008-03-18	Abbott Laboratories	Azacyclosteroid histamine-3 receptor ligands

2011
- 2011-08-19 HU HU1100453A patent/HUP1100453A2/en unknown
2012
- 2012-08-17 WO PCT/HU2012/000075 patent/WO2013027073A1/en active Application Filing

Also Published As

Publication number	Publication date
WO2013027073A1 (en)	2013-02-28

Publication	Publication Date	Title
AU341034S (en)	2012-02-17	Shroud
IL227844A0 (en)	2013-09-30	Aircraft
EP2662268A4 (en)	2014-06-11	Lid-fastening structure
PL2771471T3 (en)	2017-10-31	Construct
ZA201402236B (en)	2015-03-25	Aircraft
GB201118773D0 (en)	2011-12-14	Probe
EP2717400A4 (en)	2015-09-16	Grommet
GB201412487D0 (en)	2014-08-27	Aggregates
IL213180A0 (en)	2011-10-31	Aircraft
AU338240S (en)	2011-08-24	Salad spinner
GB201116131D0 (en)	2011-11-02	Probe
EP2762327A4 (en)	2015-05-27	Multi-pen
ZA201402257B (en)	2021-05-26	Tapered structure construction
PL3034071T3 (en)	2018-05-30	New combination
EP2719552A4 (en)	2014-09-10	Attachment structure
PT2719842E (en)	2015-12-09	Framework for structural use
SG11201402471SA (en)	2014-08-28	Photocatalyst-supporting structure
GB201210616D0 (en)	2012-08-01	Repair arrangement
HUP1100453A2 (en)	2013-02-28	Carboxamides with sterane skeleton as h3 antagonists
AU340812S (en)	2012-02-09	Mixer
GB201108441D0 (en)	2011-07-06	Grommet
GB201116630D0 (en)	2011-11-09	Reinforcement
GB201100188D0 (en)	2011-02-23	Structural members
GB201122074D0 (en)	2012-02-01	Manual Laundrey Washer
GB201209194D0 (en)	2012-07-04	Snug screen

Legal Events

Date	Code	Title	Description
2017-03-28	FA9A	Lapse of provisional patent protection due to relinquishment or protection considered relinquished