JP2002509105A - Ｉｌ−８受容体アンタゴニスト - Google Patents

Ｉｌ−８受容体アンタゴニスト

Info

Publication number: JP2002509105A
Authority: JP; Japan
Prior art keywords: alkyl; optionally substituted; heteroaryl; aryl; heterocyclic
Prior art date: 1998-01-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Withdrawn

Application number

JP2000539842A

Other languages

English (en)

Japanese (ja)

Inventor

デボラ・リン・ブライアン

キャサリン・エル・ウィドーソン

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

SmithKline Beecham Corp

Original Assignee

SmithKline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-01-16

Filing date

1999-01-15

Publication date

2002-03-26

1999-01-15 Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp

2002-03-26 Publication of JP2002509105A publication Critical patent/JP2002509105A/ja

Status Withdrawn legal-status Critical Current

Links

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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Rheumatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pulmonology (AREA)
Neurology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Dermatology (AREA)
Tropical Medicine & Parasitology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Virology (AREA)
Hematology (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Transplantation (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

JP2000539842A 1998-01-16 1999-01-15 Ｉｌ−８受容体アンタゴニスト Withdrawn JP2002509105A (ja)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US7165398P	1998-01-16	1998-01-16
US60/071,653		1998-01-16
PCT/US1999/001029 WO1999036069A1 (fr)	1998-01-16	1999-01-15	Antagonistes des recepteurs de l'interleukine-8

Publications (1)

Publication Number	Publication Date
JP2002509105A true JP2002509105A (ja)	2002-03-26

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ID=22102724

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JP2000539842A Withdrawn JP2002509105A (ja)	1998-01-16	1999-01-15	Ｉｌ−８受容体アンタゴニスト

Country Status (5)

Country	Link
EP (1)	EP1039903A4 (fr)
JP (1)	JP2002509105A (fr)
AU (1)	AU2234199A (fr)
CA (1)	CA2318195A1 (fr)
WO (1)	WO1999036069A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AR008331A1 (es) *	1997-01-23	1999-12-29	Smithkline Beecham Corp	Compuestos antagonistas de un receptor de il-8, uso de los mismos para la fabricacion de medicamentos, procedimiento para su obtencion, composicionesfarmaceuticas que los contienen
PE20011124A1 (es)	2000-03-31	2001-10-28	Upjohn Co	Nuevos agentes antibacterianos de benzosultam oxazolidinona
DE10038709A1 (de) *	2000-08-09	2002-02-28	Aventis Pharma Gmbh	Substituierte und unsubstituierte Benzooxathiazole sowie daraus abgeleitete Verbindungen
WO2003087072A1 (fr) *	2002-03-29	2003-10-23	Mochida Pharmaceutical Co., Ltd.	Agent therapeutique destine a des troubles endotheliaux
TW200418812A (en)	2002-10-29	2004-10-01	Smithkline Beecham Corp	IL-8 receptor antagonists
NZ572069A (en)	2006-04-21	2011-09-30	Smithkline Beecham Corp	IL-8 RECEPTOR ANTAGONIST N-[4-chloro-2-hydroxy-3-(3-piperidinylsulfonyl)-phenyl]-N'-(3-fluoro-2-methylphenyl)urea
CA2650007A1 (fr)	2006-04-21	2007-11-01	Smithkline Beecham Corporation	Antagonistes du recepteur de l'il-8

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3302125A1 (de) *	1983-01-22	1984-07-26	Boehringer Ingelheim KG, 6507 Ingelheim	Aminosaeure-derivate, verfahren zu ihrer herstellung und verwendung
US5504095A (en) *	1990-09-19	1996-04-02	Pfizer Inc.	Aminobenzosultam derivatives as lipoxygenase inhibitors
TR199802695T2 (xx) *	1996-06-27	1999-04-21	Smithkline Beecham Corporation	IL-8 Resept�r kar��tlar�

1999
- 1999-01-15 CA CA002318195A patent/CA2318195A1/fr not_active Abandoned
- 1999-01-15 EP EP99902334A patent/EP1039903A4/fr not_active Withdrawn
- 1999-01-15 AU AU22341/99A patent/AU2234199A/en not_active Abandoned
- 1999-01-15 WO PCT/US1999/001029 patent/WO1999036069A1/fr not_active Application Discontinuation
- 1999-01-15 JP JP2000539842A patent/JP2002509105A/ja not_active Withdrawn

Also Published As

Publication number	Publication date
WO1999036069A1 (fr)	1999-07-22
CA2318195A1 (fr)	1999-07-22
EP1039903A4 (fr)	2001-12-05
AU2234199A (en)	1999-08-02
EP1039903A1 (fr)	2000-10-04

Publication	Publication Date	Title
US6297265B2 (en)	2001-10-02	Benzoisothiazole-substituted compounds useful as IL-8 receptor antagonists
US6043374A (en)	2000-03-28	Benzisothiazolidine Compounds
JP2000513360A (ja)	2000-10-10	Ｉｌ―８レセプターアンタゴニスト
JP2004509070A (ja)	2004-03-25	Ｉｌ−８受容体アンタゴニスト
JP2001512096A (ja)	2001-08-21	Ｉｌ−８レセプターアンタゴニスト
JP2004520412A (ja)	2004-07-08	Ｉｌ−８受容体アンタゴニスト
JP2003501463A (ja)	2003-01-14	Ｉｌ−８受容体アンタゴニスト
US6316478B1 (en)	2001-11-13	IL-8 receptor antagonists
JP2003527360A (ja)	2003-09-16	Ｉｌ−８受容体アンタゴニスト
EP0971908B1 (fr)	2004-06-30	Antagoniste de recepteurs d'il-8
JP2002509105A (ja)	2002-03-26	Ｉｌ−８受容体アンタゴニスト
EP1558259B1 (fr)	2011-04-06	Dérivés de l'urée en tant qu'antagonistes du récepteur IL-8
US6436927B1 (en)	2002-08-20	IL-8 receptor antagonists
JP2002509106A (ja)	2002-03-26	Ｉｌ−８受容体アンタゴニスト
KR20020091130A (ko)	2002-12-05	Ｉｌ-８ 수용체 길항제
JP2003530328A (ja)	2003-10-14	Ｉｌ−８受容体アンタゴニスト
US20030225125A1 (en)	2003-12-04	IL-8 receptor antagonists
JP2003501450A (ja)	2003-01-14	Ｉｌ−８受容体アンタゴニスト
JP2002521368A (ja)	2002-07-16	Ｉｌ−８受容体アンタゴニスト
JP2003527361A (ja)	2003-09-16	Ｉｌ−８受容体アンタゴニスト
JP2002518300A (ja)	2002-06-25	Ｉｌ−８受容体アンタゴニスト
JP2003501470A (ja)	2003-01-14	Ｉｌ−８受容体アンタゴニスト
JP2003501471A (ja)	2003-01-14	Ｉｌ−８受容体アンタゴニスト
CZ2001270A3 (cs)	2001-07-11	Antagonista receptoru IL-8
HK1028730B (en)	2006-06-23	Il-8 receptor antagonists

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