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WO1992017066A1 - Salicylamides substitues, agent phytosanitaires - Google Patents

Salicylamides substitues, agent phytosanitaires Download PDF

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Publication number
WO1992017066A1
WO1992017066A1 PCT/EP1992/000571 EP9200571W WO9217066A1 WO 1992017066 A1 WO1992017066 A1 WO 1992017066A1 EP 9200571 W EP9200571 W EP 9200571W WO 9217066 A1 WO9217066 A1 WO 9217066A1
Authority
WO
WIPO (PCT)
Prior art keywords
hydrogen
chain
straight
carbon atoms
halogen
Prior art date
Application number
PCT/EP1992/000571
Other languages
German (de)
English (en)
Inventor
Michael Haug
Klaus Jelich
Heinz-Wilhem Dehne
Stefan Dutzmann
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Priority to BR9205820A priority Critical patent/BR9205820A/pt
Priority to JP4506350A priority patent/JPH06509320A/ja
Publication of WO1992017066A1 publication Critical patent/WO1992017066A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/36—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a singly bound oxygen or sulfur atom attached to the same carbon skeleton, this oxygen or sulfur atom not being a member of a carboxylic group or of a thio analogue, or of a derivative thereof, e.g. hydroxy-carboxylic acids
    • A01N37/38—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a singly bound oxygen or sulfur atom attached to the same carbon skeleton, this oxygen or sulfur atom not being a member of a carboxylic group or of a thio analogue, or of a derivative thereof, e.g. hydroxy-carboxylic acids having at least one oxygen or sulfur atom attached to an aromatic ring system
    • A01N37/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a singly bound oxygen or sulfur atom attached to the same carbon skeleton, this oxygen or sulfur atom not being a member of a carboxylic group or of a thio analogue, or of a derivative thereof, e.g. hydroxy-carboxylic acids having at least one oxygen or sulfur atom attached to an aromatic ring system having at least one carboxylic group or a thio analogue, or a derivative thereof, and one oxygen or sulfur atom attached to the same aromatic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/58—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/64—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/57—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and carboxyl groups, other than cyano groups, bound to the carbon skeleton

Definitions

  • R 4 represents hydrogen, alkanoyl, or an equivalent of an inorganic or organic cation
  • R 3 represents hydrogen, chlorine, bromine or methyl
  • R 4 represents hydrogen, acetyl, or an equivalent of a sodium, potassium, calcium or ammonium cation and
  • Ar represents phenyl which is monosubstituted to trisubstituted by identical or different substituents, the following being suitable as substituents:
  • R 2 represents hydrogen or trifluoromethyl
  • R 3 represents hydrogen
  • R 4 represents hydrogen, acetyl, a sodium cation
  • Ar represents phenyl which is monosubstituted or disubstituted, identically or differently, the following being suitable as substituents: fluorine, chlorine, bromine, cyano, nitro, methyl, ethyl, n- or i-propyl, n-, i-, s- or t-butyl, methoxy, ethoxy, n or i-propoxy, n-, i-, s- or t-butoxy, methylthio, ethylthio, trifluoromethyl, trifluoromethoxy, trifluoromethylthio, methoxycarbonyl or ethoxycarbonyl.
  • R 4 represents hydrogen, alkanoyl or an equivalent of an inorganic or organic cation
  • R 2-1 represents trifluoromethyl
  • R 1 , R 1-1 or R 2-1 , R 3 and R 4 have the meaning given above, with anilines of the formula (IIIa),
  • Drechslera (Conidial form: Drechslera, Syn: Helminthosporium);
  • Emulsifier 0.3 parts by weight of alkyl aryl polyglycol ether

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

On utilise pour combattre des parasites des salicylamides partiellement connus ayant la formule générale (I), dans laquelle Ar, R1, R2, R3 et R4 ont la notation donnée dans la description. L'invention concerne également de nouveaux composés ayant la formule (I) et leur préparation.
PCT/EP1992/000571 1991-03-30 1992-03-17 Salicylamides substitues, agent phytosanitaires WO1992017066A1 (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
BR9205820A BR9205820A (pt) 1991-03-30 1992-03-17 Salicilamidas substituidas, agente contra doenças de plantas
JP4506350A JPH06509320A (ja) 1991-03-30 1992-03-17 置換サリチルアミド類、植物の病気に対する薬剤

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19914110483 DE4110483A1 (de) 1991-03-30 1991-03-30 Substituierte salicylamide, mittel gegen pflanzenkrankheiten
DEP4110483.8 1991-03-30

Publications (1)

Publication Number Publication Date
WO1992017066A1 true WO1992017066A1 (fr) 1992-10-15

Family

ID=6428555

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP1992/000571 WO1992017066A1 (fr) 1991-03-30 1992-03-17 Salicylamides substitues, agent phytosanitaires

Country Status (8)

Country Link
EP (1) EP0586386A1 (fr)
JP (1) JPH06509320A (fr)
AU (1) AU1562492A (fr)
BR (1) BR9205820A (fr)
DE (1) DE4110483A1 (fr)
HU (1) HUT65081A (fr)
PL (1) PL294002A1 (fr)
WO (1) WO1992017066A1 (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996005170A1 (fr) * 1994-08-11 1996-02-22 Bayer Aktiengesellschaft 4-trifluoromethylbenzamides et leur utilisation sous forme de pesticides dans la protection phytosanitaire et la protection des materiaux
WO2003066613A1 (fr) * 2002-02-07 2003-08-14 Novartis Ag Derives de n-phenyl-2-pyrimidine-amine
AU2007203463B2 (en) * 2002-02-07 2010-12-23 Novartis Pharma Ag N-phenyl-2-pyrimidine-amine derivatives

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1035772A4 (fr) * 1997-12-04 2001-03-28 Dow Agrosciences Llc Compositions fongicides, procedes correspondants, composes et procedes concourant a leur elaboration
US6333432B1 (en) 1999-05-04 2001-12-25 Gina M. Fitzpatrick Fungicidal compositions and methods, and compounds and methods for the preparation thereof

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2967194A (en) * 1958-05-15 1961-01-03 Pennsalt Chemicals Corp 4-trifluoromethylsalicylamides
FR1318207A (fr) * 1961-03-25 1963-02-15 Cassella Farbwerke Mainkur Ag Arylamides d'acides salicyliques et leur procédé de préparation
GB1079177A (en) * 1963-06-11 1967-08-16 Stecker Internat S P A Improvements in pesticide composition for destroying internal worm parasites in animals
US3577550A (en) * 1968-05-02 1971-05-04 Dow Chemical Co N-(phenoxy)phenyl-salicylamides and their utilization as molluscidides
US3646199A (en) * 1967-07-26 1972-02-29 Ciba Ltd Salicyclic acid o-hydroxyphenylamides for combating bacteria and fungi
FR2182881A1 (fr) * 1972-03-21 1973-12-14 Hoechst Ag
US3914418A (en) * 1971-09-02 1975-10-21 Merck & Co Inc Methods of controlling liver fluke infections

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2967194A (en) * 1958-05-15 1961-01-03 Pennsalt Chemicals Corp 4-trifluoromethylsalicylamides
FR1318207A (fr) * 1961-03-25 1963-02-15 Cassella Farbwerke Mainkur Ag Arylamides d'acides salicyliques et leur procédé de préparation
GB1079177A (en) * 1963-06-11 1967-08-16 Stecker Internat S P A Improvements in pesticide composition for destroying internal worm parasites in animals
US3646199A (en) * 1967-07-26 1972-02-29 Ciba Ltd Salicyclic acid o-hydroxyphenylamides for combating bacteria and fungi
US3577550A (en) * 1968-05-02 1971-05-04 Dow Chemical Co N-(phenoxy)phenyl-salicylamides and their utilization as molluscidides
US3914418A (en) * 1971-09-02 1975-10-21 Merck & Co Inc Methods of controlling liver fluke infections
FR2182881A1 (fr) * 1972-03-21 1973-12-14 Hoechst Ag

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
CHEMICAL ABSTRACTS, vol. 87, no. 1, 4. Juli 1977, Columbus, Ohio, US; abstract no. 5662Y, H.UMEZAWA ET. AL.: 'Benzanilide derivatives' Seite 5657 ; *
CHEMICAL ABSTRACTS, vol. 88, no. 9, 27. Februar 1978, Columbus, Ohio, US; abstract no. 58568Z, H.UMEZAWA ET. AL.: 'Benzanilide derivatives as allergy and inflammation inhibitors' Seite 52 ; *
JOURNAL OF MEDICINAL CHEMISTRY. Bd. 33, Nr. 1, 1990, WASHINGTON US Seiten 136 - 142; D.L.SELWOOD ET. AL.: 'Structure-Activity Relationships of Antifilarial Antimycin Analogues: A Multivariate Pattern Recognition Study' *

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996005170A1 (fr) * 1994-08-11 1996-02-22 Bayer Aktiengesellschaft 4-trifluoromethylbenzamides et leur utilisation sous forme de pesticides dans la protection phytosanitaire et la protection des materiaux
WO2003066613A1 (fr) * 2002-02-07 2003-08-14 Novartis Ag Derives de n-phenyl-2-pyrimidine-amine
AU2003244444B9 (en) * 2002-02-07 2003-09-02 Novartis Pharma Ag N-phenyl-2-pyrimidine-amine derivatives
AU2003244444B2 (en) * 2002-02-07 2007-08-09 Novartis Pharma Ag N-phenyl-2-pyrimidine-amine derivatives
CN100347162C (zh) * 2002-02-07 2007-11-07 诺瓦提斯公司 N－苯基－2－嘧啶胺衍生物
US7456283B2 (en) 2002-02-07 2008-11-25 Novartis Ag N-phenyl-2-pyrimidine-amine derivatives
US7579467B2 (en) 2002-02-07 2009-08-25 Novartis Ag N-phenyl-2-pyrimidine-amine derivatives
US7816359B2 (en) 2002-02-07 2010-10-19 Novartis Ag N-phenyl-2-pyrimidine-amine derivatives
US7825247B2 (en) 2002-02-07 2010-11-02 Novartis Ag N-phenyl-2-pyrimidine-amine derivatives
AU2007203463B2 (en) * 2002-02-07 2010-12-23 Novartis Pharma Ag N-phenyl-2-pyrimidine-amine derivatives
KR101027044B1 (ko) 2002-02-07 2011-04-11 노파르티스 아게 Ｎ-페닐-2-피리미딘-아민 유도체
US9573928B2 (en) 2002-02-07 2017-02-21 Novartis Ag N-phenyl-2-pyrimidine-amine derivatives

Also Published As

Publication number Publication date
BR9205820A (pt) 1994-06-28
JPH06509320A (ja) 1994-10-20
HU9302763D0 (en) 1994-01-28
PL294002A1 (en) 1993-03-22
DE4110483A1 (de) 1992-10-01
EP0586386A1 (fr) 1994-03-16
AU1562492A (en) 1992-11-02
HUT65081A (en) 1994-04-28

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