WO2006004841A3 - Agonistes de galanine - Google Patents
Agonistes de galanine Download PDFInfo
- Publication number
- WO2006004841A3 WO2006004841A3 PCT/US2005/023122 US2005023122W WO2006004841A3 WO 2006004841 A3 WO2006004841 A3 WO 2006004841A3 US 2005023122 W US2005023122 W US 2005023122W WO 2006004841 A3 WO2006004841 A3 WO 2006004841A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- galanin agonists
- galanin
- agonists
- galmic
- seizure
- Prior art date
Links
- 102000019432 Galanin Human genes 0.000 title 1
- 101800002068 Galanin Proteins 0.000 title 1
- 239000000556 agonist Substances 0.000 title 1
- SLZIZIJTGAYEKK-CIJSCKBQSA-N molport-023-220-247 Chemical compound C([C@@H](C(=O)N[C@@H](C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=1N=CNC=1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CC=1N=CNC=1)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O)NC(=O)[C@H]1N(CCC1)C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CC=1C2=CC=CC=C2NC=1)NC(=O)CN)[C@@H](C)O)C1=CNC=N1 SLZIZIJTGAYEKK-CIJSCKBQSA-N 0.000 title 1
- 229940123935 Galanin receptor agonist Drugs 0.000 abstract 1
- 230000006399 behavior Effects 0.000 abstract 1
- 238000012048 forced swim test Methods 0.000 abstract 1
- DOHGPSDHRIKTDB-KBAHWNQNSA-N galmic Chemical compound O=C([C@@]1(C)C2=NC(=C(O2)C)C(=O)N[C@](C)(C2=NC(=C(O2)C)C(=O)N[C@@](C2=NC(=C(O2)C)C(=O)N1)(C)C(=O)N[C@@H](CCCCN)C(=O)OC)C(=O)NC1C2=CC=CC=C2C2=CC=CC=C21)NCC1CCCCC1 DOHGPSDHRIKTDB-KBAHWNQNSA-N 0.000 abstract 1
- 108010036472 galmic Proteins 0.000 abstract 1
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58437004P | 2004-06-29 | 2004-06-29 | |
US60/584,370 | 2004-06-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2006004841A2 WO2006004841A2 (fr) | 2006-01-12 |
WO2006004841A3 true WO2006004841A3 (fr) | 2006-04-13 |
Family
ID=35783332
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2005/023122 WO2006004841A2 (fr) | 2004-06-29 | 2005-06-29 | Agonistes de galanine |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2006004841A2 (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006047302A1 (fr) | 2004-10-21 | 2006-05-04 | Transtech Pharma, Inc. | Composes bissulfonamide utilises en tant qu'agonistes du galr1, compositions, et procedes d'utilisation associes |
MY198246A (en) * | 2015-10-23 | 2023-08-16 | Vifor Int Ag | Novel Ferroportin Inhibitors |
JP6831903B2 (ja) * | 2017-03-21 | 2021-02-17 | 富士フイルム株式会社 | ペプチド化合物およびその製造方法、スクリーニング用組成物、並びにペプチド化合物の選択方法 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6407136B1 (en) * | 1999-05-21 | 2002-06-18 | Ortho-Mcneil Pharmaceutical, Inc. | 1,4-dithiin and 1,4-dithiepin-1,1,4,4, tetroxide derivatives useful as antagonists of the human galanin receptor |
US6747060B2 (en) * | 2001-05-25 | 2004-06-08 | Kemia, Inc. | Non-natural galanin receptor ligands |
-
2005
- 2005-06-29 WO PCT/US2005/023122 patent/WO2006004841A2/fr active Application Filing
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6407136B1 (en) * | 1999-05-21 | 2002-06-18 | Ortho-Mcneil Pharmaceutical, Inc. | 1,4-dithiin and 1,4-dithiepin-1,1,4,4, tetroxide derivatives useful as antagonists of the human galanin receptor |
US6747060B2 (en) * | 2001-05-25 | 2004-06-08 | Kemia, Inc. | Non-natural galanin receptor ligands |
Also Published As
Publication number | Publication date |
---|---|
WO2006004841A2 (fr) | 2006-01-12 |
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