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BG103232A - Heterocyclic esters and amides - Google Patents

Heterocyclic esters and amides

Info

Publication number
BG103232A
BG103232A BG103232A BG10323299A BG103232A BG 103232 A BG103232 A BG 103232A BG 103232 A BG103232 A BG 103232A BG 10323299 A BG10323299 A BG 10323299A BG 103232 A BG103232 A BG 103232A
Authority
BG
Bulgaria
Prior art keywords
amides
heterocyclic esters
esters
immunophyline
enzimic
Prior art date
Application number
BG103232A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jia-He Li
Gregory Hamilton
Original Assignee
Gpi Nil Holdings, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gpi Nil Holdings, Inc. filed Critical Gpi Nil Holdings, Inc.
Publication of BG103232A publication Critical patent/BG103232A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D267/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D267/02Seven-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
BG103232A 1996-09-25 1999-03-10 Heterocyclic esters and amides BG103232A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/719,947 US5801187A (en) 1996-09-25 1996-09-25 Heterocyclic esters and amides
PCT/US1997/014624 WO1998013355A1 (en) 1996-09-25 1997-08-20 Heterocyclic esters and amides

Publications (1)

Publication Number Publication Date
BG103232A true BG103232A (en) 2000-05-31

Family

ID=24892040

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103232A BG103232A (en) 1996-09-25 1999-03-10 Heterocyclic esters and amides

Country Status (24)

Country Link
US (4) US5801187A (xx)
EP (1) EP0934287B1 (xx)
JP (1) JP2001502668A (xx)
KR (1) KR20000048589A (xx)
CN (1) CN1234795A (xx)
AR (1) AR009749A1 (xx)
AT (1) ATE432266T1 (xx)
AU (1) AU732194C (xx)
BG (1) BG103232A (xx)
BR (1) BR9712834A (xx)
CA (1) CA2263925A1 (xx)
CZ (1) CZ66099A3 (xx)
DE (1) DE69739422D1 (xx)
EA (1) EA199900140A1 (xx)
HU (1) HUP0000969A3 (xx)
ID (1) ID19588A (xx)
IL (1) IL128675A (xx)
NO (1) NO991433L (xx)
NZ (1) NZ334186A (xx)
PA (1) PA8438501A1 (xx)
PL (1) PL332183A1 (xx)
SK (1) SK26699A3 (xx)
WO (1) WO1998013355A1 (xx)
ZA (1) ZA977901B (xx)

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EP0934287B1 (en) 2009-05-27
NZ334186A (en) 2000-09-29
US5801187A (en) 1998-09-01
JP2001502668A (ja) 2001-02-27
EP0934287A4 (en) 2000-01-12
HUP0000969A3 (en) 2001-12-28
US6200972B1 (en) 2001-03-13
PL332183A1 (en) 1999-08-30
NO991433L (no) 1999-05-25
US6218544B1 (en) 2001-04-17
WO1998013355A1 (en) 1998-04-02
AU732194B2 (en) 2001-04-12
EP0934287A1 (en) 1999-08-11
CA2263925A1 (en) 1998-04-02
AU732194C (en) 2001-12-06
ATE432266T1 (de) 2009-06-15
NO991433D0 (no) 1999-03-24
AR009749A1 (es) 2000-05-03
KR20000048589A (ko) 2000-07-25
AU4076997A (en) 1998-04-17
IL128675A (en) 2002-08-14
US20030032635A1 (en) 2003-02-13
HUP0000969A2 (hu) 2000-10-28
EA199900140A1 (ru) 1999-10-28
SK26699A3 (en) 2000-01-18
ZA977901B (en) 1998-03-25
ID19588A (id) 1998-07-23
CZ66099A3 (cs) 1999-06-16
DE69739422D1 (de) 2009-07-09
CN1234795A (zh) 1999-11-10
BR9712834A (pt) 1999-11-16
PA8438501A1 (es) 2000-05-24
IL128675A0 (en) 2000-01-31

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