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HUP0301189A2 - Pirazolibifenilkarboxamidok, intermedierjeik, eljárás előállításukra és alkalmazásuk nemkívánatos mikroorganizmusok leküzdésére - Google Patents

Pirazolibifenilkarboxamidok, intermedierjeik, eljárás előállításukra és alkalmazásuk nemkívánatos mikroorganizmusok leküzdésére

Info

Publication number
HUP0301189A2
HUP0301189A2 HU0301189A HUP0301189A HUP0301189A2 HU P0301189 A2 HUP0301189 A2 HU P0301189A2 HU 0301189 A HU0301189 A HU 0301189A HU P0301189 A HUP0301189 A HU P0301189A HU P0301189 A2 HUP0301189 A2 HU P0301189A2
Authority
HU
Hungary
Prior art keywords
haloalkyl
alkyl
group
intermediates
preparation
Prior art date
Application number
HU0301189A
Other languages
English (en)
Inventor
Ralf Dunkel
Hans-Ludwig Elbe
Thomas Jaetsch
Karl-Heinz Kuck
Martin Kugler
Astrid Mauler-Machnik
Heiko Rieck
Ulrike Wachendorff-Neumann
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10122097A external-priority patent/DE10122097A1/de
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of HUP0301189A2 publication Critical patent/HUP0301189A2/hu
Publication of HUP0301189A3 publication Critical patent/HUP0301189A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/30—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C223/00—Compounds containing amino and —CHO groups bound to the same carbon skeleton
    • C07C223/06—Compounds containing amino and —CHO groups bound to the same carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

A találmány (I) általános képletű új pirazolilbifenilkarboxamidokra,előállítási eljárásaikra és nemkívánatos mikroorganizmusok leküzdéséretörténő alkalmazásukra vonatkozik. Az (I) általános képletben R1jelentése hidrogénatom, alkil-, halogénalkil-, benzil- vagypiridilmetilcsoport; R2 jelentése hidrogénatom vagy alkilcsoport; Xjelentése halogénatom, nitro-, ciano-, hidroxil-, karboxil-, alkil-,halogénalkil-, alkoxi-, halogénalkoxi-, alkiltio-, halogénalkiltio-,alkeniloxi-, alkiniloxi-, cikloalkil-, alkoxikarbonil-csoport vagyjelentése -C(R2)=N-OR1 általános képletű csoport; m jelentése 0-tól 3-ig terjedő egész szám, ahol X jelentése egymással azonos vagyegymástól különböző, ha m jelentése 2 vagy 3; Y jelentése halogénatom,nitro-, ciano-, hidroxil-, karboxil-, alkil-, halogénalkil-, alkoxi-,halogénalkoxi-, alkiltio-, halogénalkiltio-, alkeniloxi-, alkiniloxi-,cikloalkil-, alkoxikarbonil-csoport vagy alkoximino-alkil-csoport és njelentése 0-tól 4-ig terjedő egész szám, ahol Y egymással azonos vagyegymástól különböző csoportokat jelent, ha n jelentése 2, 3 vagy 4. Atalálmány magábafoglalja a céltermék előállítására használtintermediereket és ezek előállítását is. Ó
HU0301189A 2000-07-24 2001-07-11 Pyrazolyl biphenyl carboxamides, intermediates, preparation and use thereof for controlling undesired microorganisms HUP0301189A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10035860 2000-07-24
DE10122097A DE10122097A1 (de) 2000-07-24 2001-05-07 Pyrazolylbiphenylcarboxamide
PCT/EP2001/007990 WO2002008195A1 (de) 2000-07-24 2001-07-11 Pyrazolylbiphenylcarboxamide und deren verwendung zur bekämpfung unerwünschter mikroorganismen

Publications (2)

Publication Number Publication Date
HUP0301189A2 true HUP0301189A2 (hu) 2003-08-28
HUP0301189A3 HUP0301189A3 (en) 2003-11-28

Family

ID=26006491

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0301189A HUP0301189A3 (en) 2000-07-24 2001-07-11 Pyrazolyl biphenyl carboxamides, intermediates, preparation and use thereof for controlling undesired microorganisms

Country Status (11)

Country Link
US (2) US6992098B2 (hu)
EP (1) EP1313709A1 (hu)
JP (1) JP2004523467A (hu)
CN (1) CN1222514C (hu)
AU (1) AU2001270630A1 (hu)
BR (1) BR0112927A (hu)
HU (1) HUP0301189A3 (hu)
IL (1) IL153929A0 (hu)
MX (1) MXPA03000609A (hu)
PL (1) PL359809A1 (hu)
WO (1) WO2002008195A1 (hu)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001278480A1 (en) * 2000-07-24 2002-02-05 Bayer Crop Science Ag Biphenyl carboxamides
DE10122447A1 (de) * 2000-07-24 2002-04-18 Bayer Ag Biphenylcarboxamide
DE10136065A1 (de) * 2001-07-25 2003-02-13 Bayer Cropscience Ag Pyrazolylcarboxanilide
WO2004018461A2 (en) * 2002-08-23 2004-03-04 Pharmacia & Upjohn Company Llc Antibacterial benzoic acid derivatives
DE10258314A1 (de) 2002-12-13 2004-06-24 Bayer Cropscience Ag Biphenyloximether
GB0230155D0 (en) * 2002-12-24 2003-02-05 Syngenta Participations Ag Chemical compounds
DE10303589A1 (de) * 2003-01-29 2004-08-12 Bayer Cropscience Ag Pyrazolylcarboxanilide
DE10325439A1 (de) * 2003-05-21 2004-12-09 Bayer Cropscience Ag Iodpyrazolylcarboxanilide
CN101056858A (zh) * 2004-09-06 2007-10-17 巴斯福股份公司 防治病原性真菌的（杂）环基（硫代）羧酰苯胺
DE102005060468A1 (de) * 2005-12-17 2007-06-21 Bayer Cropscience Ag Thienylpyridylcarboxamide
WO2007071656A1 (de) * 2005-12-20 2007-06-28 Basf Aktiengesellschaft Verfahren zur bekämpfung des rostbefalls bei leguminosen
EP2662363A1 (en) 2012-05-09 2013-11-13 Bayer CropScience AG 5-Halogenopyrazole biphenylcarboxamides
KR20200040348A (ko) * 2018-10-08 2020-04-20 한국화학연구원 티오펜 카르복사미드계 유도체 및 이를 함유하는 식물 병해 방제제
CN119431246A (zh) * 2025-01-09 2025-02-14 浙江爱索拓科技有限公司 一种二氯苯环碳-14标记联苯吡菌胺及其制备方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4663341A (en) * 1984-02-16 1987-05-05 Rohm And Haas Company Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides
US4863947A (en) * 1985-01-11 1989-09-05 Rohm And Haas N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides and methods of their production
US5205854A (en) * 1988-04-13 1993-04-27 Basf Aktiengesellschaft Isoxazole(isothiazole)-5-carboxamides
DE3812225A1 (de) * 1988-04-13 1989-10-26 Basf Ag Isoxazol(isothiazol)-5-carbonsaeureamide
US5045554A (en) 1988-11-29 1991-09-03 Monsanto Company Substituted thiazoles and their use as fungicides
WO1991001311A1 (en) 1989-07-25 1991-02-07 Monsanto Company Substituted carboxanilidothiazoles and their use as fungicides
IN172842B (hu) 1990-05-17 1993-12-11 Boots Pharmaceuticals Limited
US5250532A (en) * 1991-04-11 1993-10-05 Dowelanco 3,4,N-trisubstituted-4,5-dihydro-1H-pyrazole-1-carboxamides and their use as insecticides
IL103614A (en) 1991-11-22 1998-09-24 Basf Ag Carboxamides for controlling botrytis and certain novel such compounds
US5223526A (en) 1991-12-06 1993-06-29 Monsanto Company Pyrazole carboxanilide fungicides and use
DE4231519A1 (de) 1992-09-21 1994-03-24 Basf Ag Cyclohex(en)ylcarbonsäureamide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen
DE4231517A1 (de) 1992-09-21 1994-03-24 Basf Ag Carbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen
MX9703687A (es) 1994-11-24 1997-08-30 Hoffmann La Roche Nuevas bencil pirimidinas.
DE19735224A1 (de) 1997-08-15 1999-02-18 Basf Ag Biphenylamide
DE19840322A1 (de) * 1998-09-04 2000-03-09 Bayer Ag Pyrazol-carboxanilide

Also Published As

Publication number Publication date
CN1222514C (zh) 2005-10-12
IL153929A0 (en) 2003-07-31
AU2001270630A1 (en) 2002-02-05
WO2002008195A1 (de) 2002-01-31
US20040053971A1 (en) 2004-03-18
BR0112927A (pt) 2003-07-01
PL359809A1 (en) 2004-09-06
US20050182120A1 (en) 2005-08-18
EP1313709A1 (de) 2003-05-28
US6992098B2 (en) 2006-01-31
CN1466578A (zh) 2004-01-07
MXPA03000609A (es) 2004-07-30
WO2002008195A8 (de) 2002-04-04
HUP0301189A3 (en) 2003-11-28
US7348350B2 (en) 2008-03-25
JP2004523467A (ja) 2004-08-05

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Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees