DE69606028D1 - Taxal derivate, deren herstellung und diese enthaltende pharmazeutische zusammensetzung - Google Patents

Taxal derivate, deren herstellung und diese enthaltende pharmazeutische zusammensetzung

Info

Publication number: DE69606028D1
Authority: DE; Germany
Prior art keywords: taxal; derivatives; production; pharmaceutical composition; composition containing
Prior art date: 1995-03-27
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

DE69606028T

Other languages

English (en)

Other versions

DE69606028T2 (de

Inventor

Herve Bouchard

Jean-Dominique Bourzat

Alain Commercon

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Aventis Pharma SA

Original Assignee

Rhone Poulenc Rorer SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-03-27

Filing date

1996-03-25

Publication date

2000-02-10

1995-03-27 Priority claimed from FR9503545A external-priority patent/FR2732340B1/fr

1995-12-22 Priority claimed from FR9515381A external-priority patent/FR2742754B1/fr

1996-03-25 Application filed by Rhone Poulenc Rorer SA filed Critical Rhone Poulenc Rorer SA

2000-02-10 Application granted granted Critical

2000-02-10 Publication of DE69606028D1 publication Critical patent/DE69606028D1/de

2000-08-10 Publication of DE69606028T2 publication Critical patent/DE69606028T2/de

2016-03-26 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Hematology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Epoxy Compounds (AREA)
Medicines Containing Plant Substances (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DE69606028T 1995-03-27 1996-03-25 Taxal derivate, deren herstellung und diese enthaltende pharmazeutische zusammensetzung Expired - Lifetime DE69606028T2 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR9503545A FR2732340B1 (fr)	1995-03-27	1995-03-27	Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
FR9515381A FR2742754B1 (fr)	1995-12-22	1995-12-22	Procede de preparation de taxoides
PCT/FR1996/000440 WO1996030355A1 (fr)	1995-03-27	1996-03-25	Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number	Publication Date
DE69606028D1 true DE69606028D1 (de)	2000-02-10
DE69606028T2 DE69606028T2 (de)	2000-08-10

Family

ID=26231838

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DE69604653T Expired - Lifetime DE69604653T2 (de)	1995-03-27	1996-03-25	Taxol derivate, deren herstellung und diese enthaltende pharmazeutischen zusammenstellungen
DE69606028T Expired - Lifetime DE69606028T2 (de)	1995-03-27	1996-03-25	Taxal derivate, deren herstellung und diese enthaltende pharmazeutische zusammensetzung

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
DE69604653T Expired - Lifetime DE69604653T2 (de)	1995-03-27	1996-03-25	Taxol derivate, deren herstellung und diese enthaltende pharmazeutischen zusammenstellungen

Country Status (41)

Country	Link
US (3)	US5889043A (de)
EP (2)	EP0817780B1 (de)
JP (2)	JP2941951B2 (de)
KR (2)	KR100297196B1 (de)
CN (2)	CN1152870C (de)
AP (2)	AP785A (de)
AR (1)	AR001440A1 (de)
AT (2)	ATE185562T1 (de)
AU (2)	AU703278B2 (de)
BG (2)	BG63009B1 (de)
BR (2)	BR9607930A (de)
CA (2)	CA2214321C (de)
CO (1)	CO4700576A1 (de)
CZ (2)	CZ287326B6 (de)
DE (2)	DE69604653T2 (de)
DK (2)	DK0817779T3 (de)
DZ (1)	DZ2009A1 (de)
EA (2)	EA000709B1 (de)
EE (2)	EE03608B1 (de)
ES (2)	ES2140075T3 (de)
GE (2)	GEP20002211B (de)
GR (2)	GR3031526T3 (de)
HU (2)	HU223732B1 (de)
IL (1)	IL117636A (de)
IS (2)	IS2058B (de)
MA (1)	MA23823A1 (de)
MY (1)	MY121225A (de)
NO (2)	NO316379B1 (de)
NZ (2)	NZ304901A (de)
OA (2)	OA10514A (de)
PE (1)	PE51097A1 (de)
PL (2)	PL188284B1 (de)
PT (1)	PT817779E (de)
RO (2)	RO115878B1 (de)
SK (2)	SK281927B6 (de)
TN (1)	TNSN96043A1 (de)
TR (2)	TR199701042T1 (de)
TW (1)	TW394765B (de)
UY (2)	UY24192A1 (de)
WO (2)	WO1996030356A1 (de)
ZA (1)	ZA962399B (de)

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FR2771092B1 (fr) *	1997-11-18	1999-12-17	Rhone Poulenc Rorer Sa	Procede de preparation de derives de la classe des taxoides
US6346543B1 (en) *	1998-08-17	2002-02-12	Aventis Pharma S.A.	Use of a taxoid to treat abnormal cell proliferation in the brain
EP0982027A1 (de) *	1998-08-17	2000-03-01	Aventis Pharma S.A.	Taxoid-Derivaten zur Behandlung von abnormaler Zellvermehrung des Gehirns
HUP0104000A3 (en) *	1998-08-20	2003-01-28	Aventis Pharma Sa	New use of taxoid derivatives
EP0982028A1 (de) *	1998-08-20	2000-03-01	Aventis Pharma S.A.	Neue Verwendung von Taxoidverbindungen
EP1020188A1 (de) *	1999-01-13	2000-07-19	Aventis Pharma S.A.	Neue Verwendung von Taxoid-Derivaten
US6649632B2 (en) *	2000-02-02	2003-11-18	Fsu Research Foundation, Inc.	C10 ester substituted taxanes
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WO2002024178A2 (en) *	2000-09-22	2002-03-28	Bristol-Myers Squibb Company	Method for reducing toxicity of combined chemotherapies
US6593334B1 (en)	2002-05-02	2003-07-15	The University Of North Carolina At Chapel Hill	Camptothecin-taxoid conjugates as antimitotic and antitumor agents
PT1534340E (pt)	2002-09-06	2012-03-13	Cerulean Pharma Inc	Polímeros à base de ciclodextrina para a administração de medicamentos ligados por ligação covalente
AU2003291458A1 (en) *	2002-11-08	2004-06-03	Bristol-Myers Squibb Company	Pharmaceutical compositions and methods of using taxane derivatives
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US20060189679A1 (en) *	2005-02-14	2006-08-24	Florida State University Research Foundation, Inc.	C10 cyclopropyl ester substituted taxane compositions
PL1871753T3 (pl)	2005-03-31	2012-12-31	Accord Healthcare Inc	Wytwarzanie taksanów z 9-dihydro-13-acetylobakatyny iii
ES2435724T3 (es) *	2005-11-04	2013-12-23	Accord Healthcare Inc.	Nuevos métodos para la preparación de taxanos usando auxiliares quirales
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1996
- 1996-03-08 MA MA24180A patent/MA23823A1/fr unknown
- 1996-03-19 PE PE1996000181A patent/PE51097A1/es not_active IP Right Cessation
- 1996-03-24 IL IL11763696A patent/IL117636A/en active Protection Beyond IP Right Term
- 1996-03-25 AU AU52781/96A patent/AU703278B2/en not_active Ceased
- 1996-03-25 CN CNB961928840A patent/CN1152870C/zh not_active Expired - Fee Related
- 1996-03-25 EA EA199700270A patent/EA000709B1/ru not_active IP Right Cessation
- 1996-03-25 EE EE9700315A patent/EE03608B1/xx unknown
- 1996-03-25 WO PCT/FR1996/000441 patent/WO1996030356A1/fr not_active Application Discontinuation
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1998
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2000
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Also Published As

Publication number	Publication date
SK281927B6 (sk)	2001-09-11
CN1179776A (zh)	1998-04-22
AU5278096A (en)	1996-10-16
EE9700323A (et)	1998-06-15
DK0817779T3 (da)	2000-06-19
MA23823A1 (fr)	1996-10-01
BR9607930A (pt)	1998-06-02
HUP9801204A3 (en)	2000-12-28
NO973923L (no)	1997-08-26
ES2143187T3 (es)	2000-05-01
EA199700269A1 (ru)	1998-04-30
US5889043A (en)	1999-03-30
WO1996030355A1 (fr)	1996-10-03
HUP9801201A2 (hu)	2000-05-28
NZ304900A (en)	1998-09-24
EE9700315A (et)	1998-06-15
JPH11502531A (ja)	1999-03-02
OA10514A (fr)	2002-04-22
OA10513A (fr)	2002-04-22
JPH11500141A (ja)	1999-01-06
NO973923D0 (no)	1997-08-26
NO973922L (no)	1997-08-26
TNSN96043A1 (fr)	2005-03-15
CN1152870C (zh)	2004-06-09
TW394765B (en)	2000-06-21
CZ287468B6 (en)	2000-12-13
EP0817780B1 (de)	1999-10-13
DK0817780T3 (da)	2000-03-27
PE51097A1 (es)	1997-12-22
IL117636A0 (en)	1996-07-23
AU711227B2 (en)	1999-10-07
UY24370A1 (es)	2001-10-25
GEP20002211B (en)	2000-08-25
NO973922D0 (no)	1997-08-26
DE69604653D1 (de)	1999-11-18
RO115878B1 (ro)	2000-07-28
EE03608B1 (et)	2002-02-15
KR19980703357A (ko)	1998-10-15
NO316379B1 (no)	2004-01-19
PL188987B1 (pl)	2005-05-31
CA2214321C (fr)	2008-01-22
KR100297196B1 (ko)	2001-11-22
MY121225A (en)	2006-01-28
CN1179775A (zh)	1998-04-22
GEP20002188B (en)	2000-07-25
PL322499A1 (en)	1998-02-02
PT817779E (pt)	2000-04-28
AP9701093A0 (en)	1997-10-31
AU5278196A (en)	1996-10-16
TR199701040T1 (xx)	1998-01-21
TR199701042T1 (xx)	1998-01-21
BG101917A (en)	1998-10-30
AP9701090A0 (en)	1997-10-31
JP2941951B2 (ja)	1999-08-30
ZA962399B (en)	1996-10-01
SK130297A3 (en)	1998-03-04
AR001440A1 (es)	1997-10-22
BG63009B1 (bg)	2001-01-31
PL188284B1 (pl)	2005-01-31
AU703278B2 (en)	1999-03-25
BR9607929A (pt)	1998-06-02
BG63121B1 (bg)	2001-04-30
JP3790826B2 (ja)	2006-06-28
NZ304901A (en)	1998-12-23
HU223732B1 (hu)	2004-12-28
US6387946B1 (en)	2002-05-14
MX9706568A (es)	1997-11-29
MX9706278A (es)	1997-10-31
IS2058B (is)	2005-10-14
CA2214321A1 (fr)	1996-10-03
AP753A (en)	1999-07-21
DE69604653T2 (de)	2000-05-31
RO115877B1 (ro)	2000-07-28
ATE188471T1 (de)	2000-01-15
SK281928B6 (sk)	2001-09-11
CA2214319C (fr)	2004-02-17
CZ287326B6 (en)	2000-10-11
SK130197A3 (en)	1998-04-08
EP0817779A1 (de)	1998-01-14
IL117636A (en)	2004-08-31
ES2140075T3 (es)	2000-02-16
CZ303297A3 (cs)	1998-01-14
UY24192A1 (es)	1996-06-14
IS4536A (is)	1997-07-31
HU223666B1 (hu)	2004-11-29
PL322465A1 (en)	1998-02-02
KR100485309B1 (ko)	2005-10-12
GR3031526T3 (en)	2000-01-31
CN1213042C (zh)	2005-08-03
EE03609B1 (et)	2002-02-15
NO316607B1 (no)	2004-03-08
EP0817780A1 (de)	1998-01-14
KR19980703287A (ko)	1998-10-15
BG101918A (en)	1998-10-30
CA2214319A1 (fr)	1996-10-03
DZ2009A1 (fr)	2002-10-23
EA000567B1 (ru)	1999-12-29
AP785A (en)	1999-11-26
WO1996030356A1 (fr)	1996-10-03
DE69606028T2 (de)	2000-08-10
ATE185562T1 (de)	1999-10-15
IS4567A (is)	1997-09-23
GR3032316T3 (en)	2000-04-27
HUP9801201A3 (en)	2000-12-28
CO4700576A1 (es)	1998-12-29
EA000709B1 (ru)	2000-02-28
CZ303097A3 (cs)	1998-01-14
EP0817779B1 (de)	2000-01-05
IS2056B (is)	2005-10-14
EA199700270A1 (ru)	1998-02-26
US20020038038A1 (en)	2002-03-28
HUP9801204A1 (hu)	2000-05-28
US6331635B1 (en)	2001-12-18

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Date	Code	Title	Description
2001-01-25	8364	No opposition during term of opposition
2002-05-29	8327	Change in the person/name/address of the patent owner	Owner name: AVENTIS PHARMA S.A., ANTONY, FR
2006-10-26	8328	Change in the person/name/address of the agent	Representative=s name: PFENNING MEINIG & PARTNER GBR, 80339 MUENCHEN
2009-07-30	8328	Change in the person/name/address of the agent	Representative=s name: MAIWALD PATENTANWALTSGESELLSCHAFT MBH, 80335 MUENC